|Description||Zopolrestat is an inhibitor of Aldose Reductase(AR). It has been shown to play roles in inflammation and cancer. It is used for the treatment of diabetic nephropathy and cardiac disease. It was developed by Pfizer and was terminated in clinic phase 2 trials.|
|B0084-358923||25 mg||$198||In stock|
|B0084-358923||50 mg||$298||In stock|
|Appearance||Off white to light brown powder|
|Synonyms||3-[(5-Trifluoromethyl-2-benzothiazolyl)methyl]-3,4-dihydro-4-oxophthalazine-1-acetic acid;CP-73850;3,4-Dihydro-4-oxo-3-[[5-(trifluoromethyl)-2-benzothiazolyl]methyl]-1-phthalazineacetic acid;Alond;Xedia;2-[4-Oxo-3-[[5-(trifluoromethyl)-1,3-benzothiazol-2-yl]methyl]phthalazin-1-yl]acetic acid;CP73850|
|Solubility||DMSO: ≥20 mg/mL|
|Application||Zopolrestat is used for the treatment of diabetic nephropathy and cardiac disease.|
|Quality Standard||In-house standard|
|Shelf Life||2 month in rt, long time|
|Quantity||Grams to Kilograms|
|Boiling Point||598.7±60.0 °C | Condition: Press: 760 Torr|
|Melting Point||197-198 °C|
|Density||1.58±0.1 g/cm3 | Condition: Temp: 20 °C Press: 760 Torr|
|Current Developer||Zopolrestat was developed by Pfizer and was terminated in clinic phase 2 trials.|
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