Z-Cyclopentyl-AP4 - CAS 103439-17-4
Category: Inhibitor
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Molecular Formula:
C6H12NO5P
Molecular Weight:
209.14
COA:
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Targets:
mGluR
Description:
Z-Cyclopentyl-AP4 is a group III mGlu receptor agonist with higher potency at mGlu4 than mGlu8 (EC50 = 49 and 124 μM, respectively). Z-Cyclopentyl-AP4 selectively inhibits synaptic activity in the lateral perforant pathway (IC50 = 130 and 1859 μM in the lateral and medial perforant pathways, respectively).
Brife Description:
group III mGlu receptor agonist
Purity:
≥98% by HPLC
Synonyms:
cis-(±)-1-Amino-3-phosphonocyclopentane carboxylic acid
MSDS:
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InChIKey:
GLBQBTFFQHNHGC-RPBIHNRISA-N
InChI:
InChI=1S/2C6H12NO5P/c2*7-6(5(8)9)2-1-4(3-6)13(10,11)12/h2*4H,1-3,7H2,(H,8,9)(H2,10,11,12)/t2*4-,6+/m10/s1
Canonical SMILES:
C1CC(CC1P(=O)(O)O)(C(=O)O)N.C1CC(CC1P(=O)(O)O)(C(=O)O)N
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Chemical Structure

CAS 103439-17-4 Z-Cyclopentyl-AP4

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