VU6001221 - CAS 2002495-17-0
Category: Inhibitor
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Molecular Formula:
Molecular Weight:
VU6001221 is a choline transporter (CHT) inhibitor (IC50 value of 270 nM) with comparable potency for choline uptake inhibition as ML352, as well as improved PK and CNS penetration. For the first time, VU6001221 allowed evaluation of a CHT inhibitor in a standard preclinical rodent cognition model, namely novel object recognition (NOR).
KEYWORDS: VU6001221 | CHT inhibitor | VU 6001221 | VU-6001221 | CAS [2002495-17-0] | Choline | CHT | Inhibitor | Proteins
Brife Description:
choline transporter (CHT) inhibitor
VU 6001221; VU-6001221
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CAS 2002495-17-0 VU6001221

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