VU6001221 - CAS 2002495-17-0
Category: Inhibitor
Please be kindly noted products are not for therapeutic use. We do not sell to patients.
Molecular Formula:
C20H26ClN3O3
Molecular Weight:
391.89
COA:
Inquire
Targets:
Others
Description:
VU6001221 is a choline transporter (CHT) inhibitor (IC50 value of 270 nM) with comparable potency for choline uptake inhibition as ML352, as well as improved PK and CNS penetration. For the first time, VU6001221 allowed evaluation of a CHT inhibitor in a standard preclinical rodent cognition model, namely novel object recognition (NOR).
KEYWORDS: VU6001221 | CHT inhibitor | VU 6001221 | VU-6001221 | CAS [2002495-17-0] | Choline | CHT | Inhibitor | Proteins
Brife Description:
choline transporter (CHT) inhibitor
Purity:
98%
Synonyms:
VU 6001221; VU-6001221
MSDS:
Inquire
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

Related Products


CB 3731
(CAS: 80015-07-2)

CB 3731 can be used in fluorine-19 nuclear magnetic resonance studies of binary and ternary complexes of thymidylate synthase.

CAS 130273-87-9 15(R)-17-phenyl trinor Prostaglandin F2α isopropyl ester

15(R)-17-phenyl trinor Prostaglandin F2α
(CAS: 130273-87-9)

15(R)-17-phenyl trinor Prostaglandin F2α isopropyl ester is a potential impurity in most commercial preparations of the latanoprost bulk drug product. The IC50 ...

CAS 926281-37-0 GGsTop

GGsTop
(CAS: 926281-37-0)

GGsTop is a selective and irreversible γ-glutamyl transpeptidase (GGT) inhibitor that inhibits GGT activation and blocks oxidative stress. Study shows that GGsT...

CI 972
(CAS: 115787-68-3)

This active molecular is a potent purine nucleoside phosphorylase inhibitor and a T cell-selective immunosuppressive agent. CI-972 inhibited proliferation of hu...

CAS 15790-91-7 (Z)-2-decenoic acid

(Z)-2-decenoic acid
(CAS: 15790-91-7)

Microorganisms commonly accumulate at interfaces as part of biofilms held together by a matrix of hydrated extracellular polymeric substances. cis-2-Decenoic ac...

CAS 129558-76-5 Tolfenpyrad

Tolfenpyrad
(CAS: 129558-76-5)

Tolfenpyrad is used as foliar insecticide for the control of green peach aphids in broccoli.

LY-183648
(CAS: 102993-90-8)

LY-183648 has antiestrogenic activity. It inhibited PAIII metastasis to the gluteal and iliac lymph nodes.

MMV390048
(CAS: 1314883-11-8)

MMV390048 is a novel antimalarial compound and it can competitively inhibit the binding of only a single protein, P. falciparum PI4 kinase, to the beads. MV3900...

Chemical Structure

CAS 2002495-17-0 VU6001221

Quick Inquiry

Verification code

Featured Items