VU 0285683 - CAS 327056-22-4
Category: Inhibitor
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Molecular Formula:
C14H7FN4O
Molecular Weight:
266.23
COA:
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Targets:
mGluR
Description:
VU 0285683 is a negative allosteric modulator of mGlu5 receptors with high affinity for the MPEP binding site. VU 0285683 exhibits anxiolytic activity in rodent models of anxiety.
Brife Description:
negative allosteric modulator of mGlu5 receptors
Purity:
≥98% by HPLC
Synonyms:
VU0285683, VU 0285683, VU-0285683; 3-Fluoro-5-[3-(2-pyridinyl)-1,2,4-oxadiazol-5-yl]-benzonitrile
MSDS:
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InChIKey:
GELAFISMURFRCA-UHFFFAOYSA-N
InChI:
InChI=1S/C14H7FN4O/c15-11-6-9(8-16)5-10(7-11)14-18-13(19-20-14)12-3-1-2-4-17-12/h1-7H
Canonical SMILES:
C1=CC=NC(=C1)C2=NOC(=N2)C3=CC(=CC(=C3)C#N)F
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Chemical Structure

CAS 327056-22-4 VU 0285683

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