UPF 1069 - CAS 1048371-03-4
Catalog number: 1048371-03-4
Category: Inhibitor
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Molecular Formula:
C17H13NO3
Molecular Weight:
279.29
COA:
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Targets:
PARP
Description:
UPF 1069 is a selective PARP2 inhibitor with IC50 of 0.3 μM. It is ~27-fold selective against PARP1.PARP activity is evaluated by utilizing commercially available recombinant bovine PARP-1 and mouse PARP-2. Briefly
Purity:
>98%
Synonyms:
UPF-1069, UPF1069, UPF 1069
MSDS:
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InChIKey:
JJWMRRNGWSITSQ-UHFFFAOYSA-N
InChI:
InChI=1S/C17H13NO3/c19-15(12-5-2-1-3-6-12)11-21-16-8-4-7-14-13(16)9-10-18-17(14)20/h1-10H,11H2,(H,18,20)
Canonical SMILES:
C1=CC=C(C=C1)C(=O)COC2=CC=CC3=C2C=CNC3=O
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Chemical Structure

CAS 1048371-03-4 UPF 1069

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