UPF 1069 - CAS 1048371-03-4
Catalog number: 1048371-03-4
Category: Inhibitor
Please be kindly noted products are not for therapeutic use. We do not sell to patients.
Molecular Formula:
C17H13NO3
Molecular Weight:
279.29
COA:
Inquire
Targets:
PARP
Description:
UPF 1069 is a selective PARP2 inhibitor with IC50 of 0.3 μM. It is ~27-fold selective against PARP1.PARP activity is evaluated by utilizing commercially available recombinant bovine PARP-1 and mouse PARP-2. Briefly
Purity:
>98%
Synonyms:
N/A
MSDS:
Inquire
InChIKey:
JJWMRRNGWSITSQ-UHFFFAOYSA-N
InChI:
InChI=1S/C17H13NO3/c19-15(12-5-2-1-3-6-12)11-21-16-8-4-7-14-13(16)9-10-18-17(14)20/h1-10H,11H2,(H,18,20)
Canonical SMILES:
C1=CC=C(C=C1)C(=O)COC2=CC=CC3=C2C=CNC3=O
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

Related PARP Products


CAS 1104546-89-5 BYK 204165

BYK 204165
(CAS: 1104546-89-5)

BYK 204165 is a potent and selective poly(ADP-ribose) polymerase (PARP)-1 inhibitor (pIC50 = 5.38 and 7.35 for PARP-2 and PARP-1, respectively). BYK 204165 is 1...

CAS 283173-50-2 Rucaparib

Rucaparib
(CAS: 283173-50-2)

Rucaparib, also named as AG-014699 or PF-01367338, is a poly (ADP ribose) polymerase (PARP) inhibitor. PARP is a DNA damage-activated nuclear enzyme that has a ...

Protease-Activated Receptor-2, amide

Protease-Activated Receptor-2, amide, also known as SLIGKV-NH2, is a highly potent protease-activated receptor-2 (PAR2) activating peptide and can also be utliz...

CAS 1038915-58-0 MK-4827 (R-enantiomer)

MK-4827 (R-enantiomer)
(CAS: 1038915-58-0)

MK-4827 (R-enantiomer) is the R form of MK-4827, which is a PARP inhibitor developed for the treatment of ovarian cancer.

CAS 344458-15-7 PJ34

PJ34
(CAS: 344458-15-7)

PJ34 is a novel and potential PARP inhibitor with potential anticancer activity. PJ34 has a high affinity for PARP-1 (IC(50) = 20 nM) .

CAS 459868-92-9 Rucaparib

Rucaparib
(CAS: 459868-92-9)

Rucaparib, also known as (AG-14699 or PF-01367338, is a tricyclic indole poly(ADP-Ribose) polymerase (PARP1) inhibitor with potential chemosensitizing, radiose...

CAS 1622262-74-1 BRCA1-IN-1

BRCA1-IN-1
(CAS: 1622262-74-1)

A novel small-molecule-like BRCA1 inhibitor (IC50= 0.53 μM) (Ki= 0.71 μM)

CAS 344458-19-1 PJ-34 HCL

PJ-34 HCL
(CAS: 344458-19-1)

PJ34 is a potent specific inhibitor of PARPl/2 with IC50 of 110 nM and 86 nM, respectively.

Chemical Structure

CAS 1048371-03-4 UPF 1069

Quick Inquiry

Verification code

Featured Items