UB 165 fumarate - CAS 200432-86-6
Category: Inhibitor
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Molecular Formula:
C13H15ClN2.C4H4O4
Molecular Weight:
350.8
COA:
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Targets:
nAChR
Description:
UB 165 fumarate is a full agonist at α3β2- and a weak partial agonist at α4β2- containing nAChRs (Ki = 0.27, 20 (IC50), 2790 and 990 nM for α4β2, α3, α7 and α1β1δε, respectively).
Brife Description:
nAChRs agonist
Purity:
≥99% by HPLC
Synonyms:
UB 165 fumarate; UB165 fumarate; UB-165 fumarate; 2-(6-Chloro-3-pyridinyl)-9-azabicyclo[4.2.1]non-2-ene fumarate
MSDS:
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InChIKey:
DZFRKSLRKAKJIB-WLHGVMLRSA-N
InChI:
InChI=1S/C13H15ClN2.C4H4O4/c14-13-7-4-9(8-15-13)11-3-1-2-10-5-6-12(11)16-10;5-3(6)1-2-4(7)8/h3-4,7-8,10,12,16H,1-2,5-6H2;1-2H,(H,5,6)(H,7,8)/b;2-1+
Canonical SMILES:
C1CC2CCC(N2)C(=C1)C3=CN=C(C=C3)Cl.C(=CC(=O)O)C(=O)O
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CAS 200432-86-6 UB 165 fumarate

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