|Description||(±)-U-50488 hydrochloride is a selective κ-opioid agonist with no μ-opioid antagonist effects. (±)-U-50488 hydrochloride blocks Na+ channels at high concentrations.|
|Brife Description||κ-opioid agonist|
|Purity||≥99% by HPLC|
|Related CAS||67198-13-4 (free base); 114528-79-9 ((-)-enantiomer); 114528-81-3 ((+)-enantiomer)|
|Synonyms||(±)-U-50488 hydrochloride; (±)-U 50488 hydrochloride; (±)-U50488 hydrochloride; trans-(±)-3,4-Dichloro-N-methyl-N-[2-(1-pyrrolidinyl)cyclohexyl]benzeneacetamide hydrochloride|
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(+)-U-50488 hydrochloride is the less active enantiomer of (±)-U-50488, which is an opioid receptor agonist.
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