TC-E 5002 - CAS 1453071-47-0
Category: Inhibitor
Please be kindly noted products are not for therapeutic use. We do not sell to patients.
Molecular Formula:
C15H27NO4
Molecular Weight:
285.38
COA:
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Targets:
Histone Demethylase
Description:
TC-E 5002 is a selective histone demethylase KDM2/7 subfamily inhibitor (IC50 = 0.2, 1.2, 6.8, 55, 83, >100 and >120 μM for KDM7A, KDM7B, KDM2A, KDM5A, KDM4C, KDM6A and KDM4A, respectively) with antitumor activity. It suppresses growth of HeLa and KYSE-150 cancer cells in vitro.
Brife Description:
histone demethylase KDM2/7 subfamily inhibitor
Purity:
≥98% by HPLC
Synonyms:
TC-E 5002; TC E 5002; TCE 5002; TCE-5002; TCE5002; TC-E-5002; N-(9-Cyclopropyl-1-oxononyl)-N-hydroxy-β-alanine
MSDS:
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InChIKey:
NEHSERYKENINRH-UHFFFAOYSA-N
InChI:
InChI=1S/C15H27NO4/c17-14(16(20)12-11-15(18)19)8-6-4-2-1-3-5-7-13-9-10-13/h13,20H,1-12H2,(H,18,19)
Canonical SMILES:
C1CC1CCCCCCCCC(=O)N(CCC(=O)O)O
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CAS 1453071-47-0 TC-E 5002

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