TC-DAPK 6 - CAS 315694-89-4
Catalog number: 315694-89-4
Category: Inhibitor
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Molecular Formula:
C17H12N2O2
Molecular Weight:
276.29
COA:
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Targets:
DAPK
Description:
An oxazalone compound that acts as a potent, ATP-competitive, and highly selective death-associated protein kinase (DAPK) inhibitor (IC50 = 69 and 225 nM against DAPK1 and DAPK3, respectively, with 10 µM ATP), while exhibiting much reduced or no activity against a panel of 48 other kinases even at concentrations as high as 10 µM.
Purity:
>98%
Synonyms:
DAPK inhibitor
MSDS:
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InChIKey:
GFGMISOSPOPSHN-QCTDOKRBSA-N
InChI:
InChI=1S/C17H12N2O2/c20-17-15(11-14-7-4-10-18-12-14)19-16(21-17)9-8-13-5-2-1-3-6-13/h1-12H/b9-8+,15-11+
Canonical SMILES:
C1=CC=C(C=C1)C=CC2=NC(=CC3=CN=CC=C3)C(=O)O2
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Chemical Structure

CAS 315694-89-4 TC-DAPK 6

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