|Description||TC 1 is a high affinity σ1 receptor ligand with selectivity over σ2 receptors (Ki = 10 and 370 nM respectively). TC 1 exhibits low affinity for dopamine (DAT), serotonin (SERT), noradrenalin (NET) transporters (Ki > 10 μM) and dopamine D2 receptors (Ki = 1226 nM).|
|Brife Description||σ1 receptor ligand|
|Purity||≥99% by HPLC|
|Synonyms||TC 1; TC1; TC-1; (N-(3'-Fluorophenyl)ethyl-4-azahexacyclo[5.4.1.02,6.03,10.05,9.08,11]dodecan-3-ol|
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