TC 1 - CAS 362512-81-0
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C19H20FNO
Molecular Weight:
297.37
COA:
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Targets:
Sigma Receptor
Description:
TC 1 is a high affinity σ1 receptor ligand with selectivity over σ2 receptors (Ki = 10 and 370 nM respectively). TC 1 exhibits low affinity for dopamine (DAT), serotonin (SERT), noradrenalin (NET) transporters (Ki > 10 μM) and dopamine D2 receptors (Ki = 1226 nM).
Brife Description:
σ1 receptor ligand
Purity:
≥99% by HPLC
Synonyms:
(N-(3'-Fluorophenyl)ethyl-4-azahexacyclo[5.4.1.02,6.03,10.05,9.08,11]dodecan-3-ol
MSDS:
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InChIKey:
FYGREZKTJIXWIH-UHFFFAOYSA-N
InChI:
InChI=1S/C19H20FNO/c20-9-3-1-2-8(6-9)4-5-21-18-14-10-7-11-13-12(10)15(18)17(13)19(21,22)16(11)14/h1-3,6,10-18,22H,4-5,7H2
Canonical SMILES:
C1C2C3C4C1C5C2C6C3C4C5(N6CCC7=CC(=CC=C7)F)O
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Chemical Structure

CAS 362512-81-0 TC 1

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