T-0201 Sodium - CAS 188307-16-6
Catalog number: 188307-16-6
Category: Inhibitor
Please be kindly noted products are not for therapeutic use. We do not sell to patients.
Molecular Formula:
C27H28BrN5NaO5S+
Molecular Weight:
637.51
COA:
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Targets:
Endothelin Receptor
Description:
The sodium salt form of T-0201 which has been found to be an Endothelin A receptor antagonist that could be used as as anti-ischaemic agent and was once studied in heart failure and pulmonary hypertension.
Purity:
98%
Appearance:
Powder
Synonyms:
T-0201 Sodium; T0201 Sodium; T 0201 Sodium; N-(6-(2-((5-bromopyrimidin-2-yl)oxy)ethoxy)-5-(p-tolyl)pyrimidin-4-yl)-4-(1-hydroxy-2-methylpropan-2-yl)benzenesulfonamide sodium salt
Storage:
Store in a cool and dry place and at 0 - 4 °C for short term (days to weeks) or -20 °C for long term (months to years).
MSDS:
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Quality Standard:
In-house standard
Quantity:
Milligram-Grams
InChIKey:
XZAJEZRCZRZIQI-UHFFFAOYSA-N
InChI:
InChI=1S/C27H28BrN5O5S.Na/c1-18-4-6-19(7-5-18)23-24(33-39(35,36)22-10-8-20(9-11-22)27(2,3)16-34)31-17-32-25(23)37-12-13-38-26-29-14-21(28)15-30-26;/h4-11,14-15,17,34H,12-13,16H2,1-3H3,(H,31,32,33,35,36);/q;+1
Canonical SMILES:
CC1=CC=C(C=C1)C2=C(N=CN=C2OCCOC3=NC=C(C=[NH+]3)Br)N=S(=O)(C4=CC=C(C=C4)C(C)(C)CO)[O-].[Na+]
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