SB 742457 hydrochloride - CAS 607742-55-2
Category: Inhibitor
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Molecular Formula:
C19H19N3O2S.HCl
Molecular Weight:
389.9
COA:
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Targets:
5-HT Receptor
Description:
SB 742457 hydrochloride is a selective 5-HT6 antagonist with >100-fold selectivity over other receptors. It is a potential agent added to stabilize donepezil treatment in subjects with mild-to-moderate Alzheimer's disease.
Brife Description:
5-HT6 antagonist
Purity:
99%
Related CAS:
607742-69-8 (free base)
Synonyms:
GSK-742457 hydrochloride; RVT-101 hydrochloride; SB-742457 hydrochloride; GSK 742457 hydrochloride; RVT 101 hydrochloride; SB 742457 hydrochloride; GSK742457 hydrochloride; RVT101 hydrochloride; SB742457 hydrochloride; Intepirdine hydrochloride; 3-Phenylsulfonyl-8-piperazin-1-yl-quinoline hydrochloride
MSDS:
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Application:
potential treatment of Alzheimer's disease in combination with donepezil
InChIKey:
BWLWNUQEZNYKAU-UHFFFAOYSA-N
InChI:
InChI=1S/C19H19N3O2S.ClH/c23-25(24,16-6-2-1-3-7-16)17-13-15-5-4-8-18(19(15)21-14-17)22-11-9-20-10-12-22;/h1-8,13-14,20H,9-12H2;1H
Canonical SMILES:
C1CN(CCN1)C2=CC=CC3=CC(=CN=C32)S(=O)(=O)C4=CC=CC=C4.Cl
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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CAS 607742-55-2 SB 742457 hydrochloride

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