[Sar9,Met(O2)11]-Substance P - CAS 110880-55-2
Category: Inhibitor
Please be kindly noted products are not for therapeutic use. We do not sell to patients.
Molecular Formula:
C64H100N18O15S
Molecular Weight:
1393.66
COA:
Inquire
Targets:
Neurokinin Receptor
Description:
A selective agonist of tachykinin NK1 receptor
Sequence:
RPKPQQFFGLX
Synonyms:
H-DL-Arg-DL-Pro-DL-Lys-DL-Pro-DL-Gln-DL-Gln-DL-Phe-DL-Phe-Sar-DL-Leu-DL-Met(O2)-NH2; RPKPQQFFGLX; DL-arginyl-DL-prolyl-DL-lysyl-DL-prolyl-DL-glutaminyl-DL-glutaminyl-DL-phenylalanyl-DL-phenylalanyl-sarcosyl-DL-leucyl-S,S-dioxo-DL-methioninamide; 2-[[1-[6-amino-2-[[1-[2-amino-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]hexanoyl]pyrrolidine-2-carbonyl]amino]-N-[5-amino-1-[[1-[[1-[[2-[[1-[(1-amino-4-methylsulfonyl-1-oxobutan-2-yl)amino]-4-methyl-1-oxopentan-2-yl]amino]-2-oxoethyl]-methylamino]-1-oxo-3-phenylpropan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]amino]-1,5-dioxopentan-2-yl]pentanediamide
Solubility:
DMSO
Storage:
Store in a cool and dry place (or refer to the Certificate of Analysis).
MSDS:
Inquire
Density:
1.43±0.1 g/cm3
InChIKey:
OUPXSLGGCPUZJJ-UHFFFAOYSA-N
InChI:
1S/C64H100N18O15S/c1-38(2)34-46(57(89)74-42(54(69)86)28-33-98(4,96)97)73-53(85)37-80(3)62(94)48(36-40-18-9-6-10-19-40)79-58(90)47(35-39-16-7-5-8-17-39)78-56(88)43(24-26-51(67)83)75-55(87)44(25-27-52(68)84)76-59(91)50-23-15-32-82(50)63(95)45(21-11-12-29-65)77-60(92)49-22-14-31-81(49)61(93)41(66)20-13-30-72-64(70)71/h5-10,16-19,38,41-50H,11-15,20-37,65-66H2,1-4H3,(H2,67,83)(H2,68,84)(H2,69,86)(H,73,85)(H,74,89)(H,75,87)(H,76,91)(H,77,92)(H,78,88)(H,79,90)(H4,70,71,72)
Canonical SMILES:
CC(C)CC(C(=O)NC(CCS(=O)(=O)C)C(=O)N)NC(=O)CN(C)C(=O)C(CC1=CC=CC=C1)NC(=O)C(CC2=CC=CC=C2)NC(=O)C(CCC(=O)N)NC(=O)C(CCC(=O)N)NC(=O)C3CCCN3C(=O)C(CCCCN)NC(=O)C4CCCN4C(=O)C(CCCN=C(N)N)N
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

Related Neurokinin Receptor Products


CAS 174636-32-9 SB 223412

SB 223412
(CAS: 174636-32-9)

SB 223412 is a brain penetrating and orally bioactive non-peptide NK3 receptor antagonist (Ki = 1, 144 and >100000 nM for human NK3, NK2 and NK1 receptors, resp...

CAS 137593-52-3 GR 64349

GR 64349
(CAS: 137593-52-3)

GR 64349 is a potent and selective agonist of tachykinin NK2 receptor (EC50 = 3.7 nM in rat colon).

CAS 264618-38-4 SSR 146977 hydrochloride

SSR 146977 hydrochloride
(CAS: 264618-38-4)

SSR 146977 hydrochloride is a potent and selective NK3 receptor antagonist (Ki = 0.26 and 19.3 nM in CHO cells expressing the human NK3 and NK2 receptor, respec...

CAS 2990-43-4 Eledoisin-Related Peptide

Eledoisin-Related Peptide
(CAS: 2990-43-4)

Eledoisin-Related Peptide is a tachykinin receptor ligand.

CAS 103222-11-3 RC 160

RC 160
(CAS: 103222-11-3)

RC 160 is a cyclic octapeptide somatostatin analog (Ki= 0.7, 5.4, 30.9, 45 and > 1000 nM for sst5, sst2, sst3, sst4 and sst1 receptors respectively). RC 160 is ...

CAS 148700-85-0 L-733,060

L-733,060
(CAS: 148700-85-0)

L-733,061, a phenylpiperidine derivative, has been found to be a NK1 receptor antagonist that could probably be antidepressant/ anxiolytic agent and also show a...

CAS 110880-55-2 [Sar9,Met(O2)11]-Substance P

[Sar9,Met(O2)11]-Substance P
(CAS: 110880-55-2)

A selective agonist of tachykinin NK1 receptor

CAS 86933-75-7 Neurokinin B

Neurokinin B
(CAS: 86933-75-7)

Neurokinin B, one of the tachykinin family of peptides, binds a family of GPCRs—including neurokinin receptor 1 (NK1R), NK2R, and NK3R to mediate their biologic...

Chemical Structure

CAS 110880-55-2 [Sar9,Met(O2)11]-Substance P

Quick Inquiry

Verification code

Featured Items