SAR 216471 hydrochloride - CAS 1279829-64-9
Category: Inhibitor
Please be kindly noted products are not for therapeutic use. We do not sell to patients.
Molecular Formula:
C28H31ClN8O3.HCl
Molecular Weight:
599.51
COA:
Inquire
Targets:
P2Y Receptor
Description:
SAR 216471 hydrochloride is a potent and reversible P2Y12 antagonist (IC50 = 17 nM), displaying antiplatelet and antithrombotic activity in vivo.
Brife Description:
P2Y12 antagonist
Purity:
≥98% by HPLC
Synonyms:
SAR 216471 hydrochloride; SAR-216471 hydrochloride; SAR216471 hydrochloride; 5-Chloro-N-[6-[5-methyl-4-(1-oxobutyl)-1H-pyrazol-1-yl]-3-pyridazinyl]-1-[2-(4-methyl-1-piperazinyl)-2-oxoethyl]-1H-indole-3-carboxamide hydrochloride
MSDS:
Inquire
InChIKey:
UQLWHBMSQKUYAI-UHFFFAOYSA-N
InChI:
InChI=1S/C28H31ClN8O3.ClH/c1-4-5-24(38)21-15-30-37(18(21)2)26-9-8-25(32-33-26)31-28(40)22-16-36(23-7-6-19(29)14-20(22)23)17-27(39)35-12-10-34(3)11-13-35;/h6-9,14-16H,4-5,10-13,17H2,1-3H3,(H,31,32,40);1H
Canonical SMILES:
CCCC(=O)C1=C(N(N=C1)C2=NN=C(C=C2)NC(=O)C3=CN(C4=C3C=C(C=C4)Cl)CC(=O)N5CCN(CC5)C)C.Cl
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

Related P2Y Receptor Products


CAS 936500-94-6 Elinogrel

Elinogrel
(CAS: 936500-94-6)

Elinogrel is a P2Y12 antagonist displaying antiplatelet activity.

CAS 367909-40-8 MRS 2279

MRS 2279
(CAS: 367909-40-8)

MRS 2279 is the first broadly applicable, selective and high affinity competitive antagonist radioligand for a P2Y receptor (Ki = 2.5 nM; IC50 = 51.6 nM).

CAS 1448858-83-0 MRS 2693 trisodium salt

MRS 2693 trisodium salt
(CAS: 1448858-83-0)

MRS 2693 trisodium salt is a selective P2Y6 agonist (EC50 = 0.015 μM at the hP2Y6 receptor), with no activity at other P2Y subtypes.

CAS 120202-66-6 Clopidogrel

Clopidogrel
(CAS: 120202-66-6)

Clopidogrel is converted to its active metabolite by cytochrome P450 (CYP) enzymes.

CAS 1047980-83-5 MRS 2768 tetrasodium salt

MRS 2768 tetrasodium salt
(CAS: 1047980-83-5)

MRS 2768 tetrasodium salt is a selective P2Y2 agonist (EC50 = 1.89 μM), with no affinity for human P2Y4 or P2Y6 receptors.

CAS 1343364-70-4 2-ThioUTP tetrasodium salt

2-ThioUTP tetrasodium salt
(CAS: 1343364-70-4)

2-ThioUTP tetrasodium salt is a potent and selective P2Y2 agonist (EC50 = 0.035, 0.35 and 1.5 μM for hP2Y2, hP2Y4 and hP2Y6 receptors, respectively).

CAS 145782-74-7 AR-C 66096 tetrasodium salt

AR-C 66096 tetrasodium salt
(CAS: 145782-74-7)

The sodium salt form of AR-C 66096, which has been found to be a P2Y12 receptor antagonist and could be probably used as an antithrombotic agent.

CAS 389574-19-0 Prasugrel Hydrochloride

Prasugrel Hydrochloride
(CAS: 389574-19-0)

Prasugrel is a platelet inhibitor (IC50=1.8 μM) , as a third-generation thienopyridine.

Chemical Structure

CAS 1279829-64-9 SAR 216471 hydrochloride

Quick Inquiry

Verification code

Featured Items