SAR 216471 hydrochloride - CAS 1279829-64-9
Category: Inhibitor
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Molecular Formula:
C28H31ClN8O3.HCl
Molecular Weight:
599.51
COA:
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Targets:
P2Y Receptor
Description:
SAR 216471 hydrochloride is a potent and reversible P2Y12 antagonist (IC50 = 17 nM), displaying antiplatelet and antithrombotic activity in vivo.
Brife Description:
P2Y12 antagonist
Purity:
≥98% by HPLC
Synonyms:
5-Chloro-N-[6-[5-methyl-4-(1-oxobutyl)-1H-pyrazol-1-yl]-3-pyridazinyl]-1-[2-(4-methyl-1-piperazinyl)-2-oxoethyl]-1H-indole-3-carboxamide hydrochloride
MSDS:
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InChIKey:
UQLWHBMSQKUYAI-UHFFFAOYSA-N
InChI:
InChI=1S/C28H31ClN8O3.ClH/c1-4-5-24(38)21-15-30-37(18(21)2)26-9-8-25(32-33-26)31-28(40)22-16-36(23-7-6-19(29)14-20(22)23)17-27(39)35-12-10-34(3)11-13-35;/h6-9,14-16H,4-5,10-13,17H2,1-3H3,(H,31,32,40);1H
Canonical SMILES:
CCCC(=O)C1=C(N(N=C1)C2=NN=C(C=C2)NC(=O)C3=CN(C4=C3C=C(C=C4)Cl)CC(=O)N5CCN(CC5)C)C.Cl
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CAS 1279829-64-9 SAR 216471 hydrochloride

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