|Description||The hydrochloride salt form of S1RA which is a σ1 receptor antagonist that has been found to have potential effect in pain therapy. It is still under Phase II clinical trial. IC50: 17 nM (Ki).|
|Synonyms||S1RA hydrochloride; S1RA (hydrochloride); E-52862 hydrochloride; E 52862 hydrochloride; E52862 hydrochloride; SCHEMBL99116; UNII-18XZ7850YN|
|Solubility||DMSO:≥ 57 mg/mL|
|Application||The hydrochloride salt form of S1RA which is a σ1 receptor antagonist that has been found to have potential effect in pain therapy.|
|Shelf Life||As supplied, 2 years from the QC date provided on the Certificate of Analysis, when stored properly|
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