(S)-H-1152 dihydrochloride - CAS 451462-58-1
Catalog number:
451462-58-1
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C16H21N3O2S
Molecular Weight:
319.42
COA:
Inquire
Targets:
ROCK
Description:
(S)-H-1152 dihydrochloride is a Rho-kinase inhibitor and cell permeable inhibitor of ROCK (Ki = 1.6 nM).
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Purity:
≥98%
Appearance:
White to off-white solid
Synonyms:
4-Methyl-5-{[(2S)-2-methyl-1,4-diazepan-1-yl]sulfonyl}isoquinoline dihydrochloride; 4-Methyl-5-{[(2S)-2-methyl-1,4-diazepan-1-yl]sulfonyl}isoquinoline dihydrochloride;
Solubility:
Soluble in DMSO
Storage:
Store at -20 °C
MSDS:
Inquire
Application:
Rho-kinase inhibitor
Quality Standard:
Enterprise Standard
Shelf Life:
As supplied, 2 years from the QC date provided on the Certificate of Analysis, when stored properly
Quantity:
Milligrams-Grams
Melting Point:
182-184 °C
InChIKey:
BFOPDSJOLUQULZ-GXKRWWSZSA-N
InChI:
1S/C16H21N3O2S.2ClH/c1-12-9-18-11-14-5-3-6-15(16(12)14)22(20,21)19-8-4-7-17-10-13(19)2;;/h3,5-6,9,11,13,17H,4,7-8,10H2,1-2H3;2*1H/t13-;;/m0../s1
Canonical SMILES:
C[C@H]1CNCCCN1S(=O)(=O)C2=CC=CC3=C2C(=CN=C3)C.Cl.Cl
Current Developer:
Nonindustrial source
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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CAS 451462-58-1 (S)-H-1152 dihydrochloride

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