(S)-6-Hydroxybuspirone hydrochloride
Category: Inhibitor
Please be kindly noted products are not for therapeutic use. We do not sell to patients.
Molecular Formula:
C21H31N5O3.HCl
Molecular Weight:
437.96
COA:
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Targets:
5-HT Receptor
Description:
A major active metabolite of Buspirone and a 5-HT1A partial agonist. In comparison with the (R)-enantiomer, (S)-6-Hydroxybuspirone hydrochloride is cleared more slowly from blood and has lower affinity and selectivity for the 5HT1A receptor.
Brife Description:
5-HT1A partial agonist
Purity:
99%
Synonyms:
BMS 442606 hydrochloride; BMS442606 hydrochloride; BMS-442606 hydrochloride; (10S)-10-hydroxy-8-[4-(4-pyrimidin-2-ylpiperazin-1-yl)butyl]-8-azaspiro[4.5]decane-7,9-dione hydrochloride
MSDS:
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InChIKey:
QQVBLEXAVSAUDT-GMUIIQOCSA-N
InChI:
InChI=1S/C21H31N5O3.ClH/c27-17-16-21(6-1-2-7-21)18(28)19(29)26(17)11-4-3-10-24-12-14-25(15-13-24)20-22-8-5-9-23-20;/h5,8-9,18,28H,1-4,6-7,10-16H2;1H/t18-;/m1./s1
Canonical SMILES:
C1CCC2(C1)CC(=O)N(C(=O)C2O)CCCCN3CCN(CC3)C4=NC=CC=N4.Cl
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