|Description||(S)-(-)-4-Amino-2-hydroxybutyric acid is an analogue of γ-aminobutyric acid (GABA) that exhibits potential inhibitory activity on GABA binding and uptake by brain.|
|B0084-091852||200 g||$198||In stock|
DMCM hydrochloride is a benzodiazepine inverse agonist exhibiting anxiogenic and potent convulsant activity.
Etomidate is a GABAA receptor agonist, used as a short-acting anaesthetic agent or sedative.
CH-50911 is a selective GABA-B antagonist with IC50 value of 1.1 μM. It is developed by Schering-Plough Corporation. CH-50911 is often used in pharmacology rese...
CGP52432 is a potent and selective GABAB receptor antagonist with IC50 value of 85 nM.
Isoguvacine hydrochloride is a selective GABA receptor agonist with anticonvulsant and antiepileptic effect, developed for Neuroscience research.
(±)-Nipecotic acid is a nonselective GAT inhibitor that also induces GABA release through a process termed 'heteroexchange. IC50 = 8, 38, 106 and 2370 μM for hG...
Flumazenil is a GABAA receptor antagonist and the only GABAA receptor antagonist on the market today.
Arbaclofen, the R-enantiomer of baclofen, is a selective gamma-amino butyric acid type B receptor agonist used for autism spectrum disorder and fragile X syndro...
Phaclofen, a phosphonic acid derivative of Baclofen, is a selective GABAB antagonist.
CP 615003 mesylate
CP 615003 mesylate is a potent and selective GABAA receptor partial agonist potentially useful in treating generalized anxiety disorder.
BAR-501, a UDCA derivative, is a selective GPBAR1 agonist devoid of any FXR agonistic activity. BAR-501 effectively transactivates GPBAR1 in HEK293 cells overex...
CGP 13501 is a positive allosteric modulator of GABAB receptors, potentiating the effects of GABA at this receptor type.
(+)-Bicuculline is a competitive antagonist of GABAA receptors with IC50 of 2 μM, also blocks Ca(2+)-activated potassium channels.
Lesogaberan is a potent and selective GABAB receptor agonist that limit the clinical use of baclofen for the treatment of GERD.
Etomidate hydrochloride is a GABAA receptor agonist used for the induction of general anaesthesia.
CGP 36216 hydrochloride
CGP 36216 hydrochloride is a selective GABAB antagonist that is active to presynaptic receptors but inactive to postsynaptic receptors.
Ocinaplon is a GABAA receptor modulator and it can be used for the treatment of generalized anxiety disorder.
(R)-baclofen a selective GABAB agonist.
Pregnenolone sulfate sodium salt
Pregnenolone sulfate, a metabolite of the natural steroid hormone pregnenolone, is a neurosteroid that has been demonstrated to antagonize the GABAA receptor ch...
GS 39783 is an allosteric positive modulator of GABAB receptors, decreases cocaine self-administration, blocks the rewarding properties of nicotine and produces...