|Description||RU-SKI 43 is a small molecule inhibitor of Hhat(Hedgehog acyltransferase) (IC50 = 0.85 µM). RU-SKI 43 is cell-permeable and inhibits both autocrine and paracrine Shh-induced activation of Gli-mediated transcription. It attenuates pancreatic cancer cell proliferation.|
|Purity||≥98% by HPLC|
|Synonyms||RU-SKI 43 hydrochloride; RU SKI 43 hydrochloride; RUSKI 43 hydrochloride; 2-((2-Methylbutyl)amino)-1-(4-((3-methylphenoxy)methyl-6,7-dihydrothieno[3,2-c]pyridin-5(4H)-yl)ethanone hydrochloride|
|Storage||Store in a cool and dry place (or refer to the Certificate of Analysis).|
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