Ribuvaptan - CAS 1245620-47-6
Catalog number: 1245620-47-6
Category: Inhibitor
Please be kindly noted products are not for therapeutic use. We do not sell to patients.
Molecular Formula:
C23H20ClF6N5O5
Molecular Weight:
595.88
COA:
Inquire
Targets:
Vasopressin Receptor
Description:
Ribuvaptan is a vasopressin receptor antagonist originated by Bayer HealthCare Pharmaceuticals. Now, Ribuvaptan is still in phase I development for the treatment of Heart failure in Germany.
Purity:
98%
Appearance:
Powder
Synonyms:
UNII-6004MB8Y0D; 6004MB8Y0D;[(2R)-2-[[2-[3-(4-chlorophenyl)-5-oxo-4-[(2S)-3,3,3-trifluoro-2-hydroxypropyl]-1,2,4-triazol-1-yl]acetyl]amino]-2-[3-(trifluoromethyl)phenyl]ethyl] carbamate
Solubility:
Soluble in DMSO
Storage:
-20°C Freezer
MSDS:
Inquire
Application:
Heart failure
Quality Standard:
In-house standard
Shelf Life:
2 month in rt, long time
Quantity:
Milligrams-Grams
InChIKey:
JYRCFPAYSZZCBP-IRXDYDNUSA-N
InChI:
nChI=1S/C23H20ClF6N5O5/c24-15-6-4-12(5-7-15)19-33-35(21(39)34(19)9-17(36)23(28,29)30)10-18(37)32-16(11-40-20(31)38)13-2-1-3-14(8-13)22(25,26)27/h1-8,16-17,36H,9-11H2,(H2,31,38)(H,32,37)/t16-,17-/m0/s1
Canonical SMILES:
C1=CC(=CC(=C1)C(F)(F)F)C(COC(=O)N)NC(=O)CN2C(=O)N(C(=N2)C3=CC=C(C=C3)Cl)CC(C(F)(F)F)O
Current Developer:
Originator:Bayer HealthCare Pharmaceuticals
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