|Description||(R)-(-)-PK 11195 is the (R)-enantiomer of PK 11195, which is a peripheral benzodiazepine antagonist with high affinity for PBR in all species. It is used as a drug reference standard of [11C](R)-PK 11195 in PET studies.|
|Brife Description||peripheral benzodiazepine antagonist|
S 12 is a survivin inhibitor that alters spindle formation, resulting in mitotic arrest (by disrupting metaphase at the G2/M stage) and apoptosis. It inhibits c...
Glafenine hydrochloride, an anthranilic acid derivative, is a non-narcotic analgesic and non-steroidal anti-inflammatory drug. It is an ABCG2 inhibitor (IC50= 3...
(±)-Lauroylcarnitine chloride is an acylcarnitine used to improve in vivo absorption of certain hydrophilic compounds.
BoNT-IN-1 is a potent inhibitor of Botulinum neurotoxin A light chain (IC50 = 0.9 uM).
Tafamidis is a potent and selective transthyretin kinetic stabilizer that inhibits the amyloid cascade. It is a drug for the amelioration of transthyretin-relat...
Eliglustat is a glucosylceramide synthase inhibitor indicated for the long-term treatment of type 1 Gaucher disease in patients who are CYP2D6 extensive metabol...
NSC134754 is a Heat Shock Factor 1 (HSF1) inhibitor. It can induce inhibition of HSF1, SP1 and NF-κB triggers the loss of the natural killer cell-activating lig...
Ginsenoside Rb2, a sort of saponin substance, is extracted from ginseng and could inhibit the tumor growth and metastasis by destructing the angiogenesis.