|Description||(R)-(-)-LY 426965 dihydrochloride is a selective 5-HT1A antagonist that is less active than its opposite (S)-(+)-enantiomer LY 426965.|
|Brife Description||5-HT1A antagonist|
|Synonyms||(R)-(-)-LY 426965 dihydrochloride; (R)-(-)-LY426965 dihydrochloride; (R)-(-)-LY-426965 dihydrochloride; (2R)-1-cyclohexyl-4-[4-(2-methoxyphenyl)piperazin-1-yl]-2-methyl-2-phenylbutan-1-one dihydrochloride|
5-HT2 antagonist 1
A potent antagonist of 5-HT2 receptor
Eptapirone, a triazine derivative, has been found to be a 5-HT1A receptor agonist and was once studied as an antidepressant agent. pKi: 8.33.
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