(R)-(-)-JQ1 - CAS 1268524-71-5
Catalog number:
1268524-71-5
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C23H25ClN4O2S
Molecular Weight:
456.99
COA:
Inquire
Targets:
BET Bromodomain
Description:
The (R) - isomer form of JQ1 which is a BET inhibitor that could probably influence the inflammatory expression at some extent.
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Purity:
95%
Appearance:
Powder
Synonyms:
1268524-71-5;(-)-JQ-1;(-)-JQ1;(R)-tert-Butyl2-(4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)acetate;SCHEMBL881208;CHEMBL3220211
Solubility:
DMSO >150 mg/mL; Water <1 mg/mL; Ethanol 125 mg/mL
Storage:
-20ºC Freeze
MSDS:
Inquire
Application:
The (R) - isomer form of JQ1 which is a BET inhibitor that could probably influence the inflammatory expression at some extent.
Shelf Life:
As supplied, 2 years from the QC date provided on the Certificate of Analysis, when stored properly
Quantity:
Milligrams-Grams
InChIKey:
DNVXATUJJDPFDM-QGZVFWFLSA-N
InChI:
InChI=1S/C23H25ClN4O2S/c1-12-13(2)31-22-19(12)20(15-7-9-16(24)10-8-15)25-17(11-18(29)30-23(4,5)6)21-27-26-14(3)28(21)22/h7-10,17H,11H2,1-6H3/t17-/m1/s1
Canonical SMILES:
CC1=C(SC2=C1C(=NC(C3=NN=C(N32)C)CC(=O)OC(C)(C)C)C4=CC=C(C=C4)Cl)C
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CAS 1268524-71-5 (R)-(-)-JQ1

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