(R)-DRF053 dihydrochloride - CAS 1241675-76-2
Category: Inhibitor
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Molecular Formula:
C23H27N7O.2HCl
Molecular Weight:
490.43
COA:
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Targets:
CDK | CK1
Description:
The hydrochloride salt form of (R)-DRF053, which is a cdk/CK1 inhibitor and could be used in studies in the cancer treatment with combinations of CDK kinase and ERK inhibitors.
Purity:
≥98% by HPLC
Appearance:
Yellow Solid
Synonyms:
2-[[9-(1-Methylethyl)-6-[[3-(2-pyridinyl)phenyl]amino]-9H-purin-2-yl]amino]-1-butanol dihydrochloride
MSDS:
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InChIKey:
BQPRBNGSDBTKAK-ZEECNFPPSA-N
InChI:
InChI=1S/C23H27N7O.2ClH/c1-4-17(13-31)27-23-28-21(20-22(29-23)30(14-25-20)15(2)3)26-18-9-7-8-16(12-18)19-10-5-6-11-24-19;;/h5-12,14-15,17,31H,4,13H2,1-3H3,(H2,26,27,28,29);2*1H/t17-;;/m1../s1
Canonical SMILES:
CCC(CO)NC1=NC2=C(C(=N1)NC3=CC=CC(=C3)C4=CC=CC=N4)N=CN2C(C)C.Cl.Cl
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CAS 1241675-76-2 (R)-DRF053 dihydrochloride

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