|Description||(R)-1,2,3,4-Tetrahydro-3-isoquinolinecarboxylic acid is a constrained Phe analogue which can fold into a beta-bend and a helical structure, and to adopt a preferred side-chain disposition in the peptide.|
EED-226 is a novel allosteric Polycomb repressive complex 2 (PRC2) inhibitor (IC50 = 23.4 nM when the substrate is H3K27me0 peptide and IC50 = 53.5 nM when the ...
Spexin is an endogenous satiety-inducing peptide and a potent galanin receptor 2/3 (GAL2/GAL3) agonist (EC50 = 45.7 and 112.2 nM, respectively), displaying no s...
This molecular is a novel non-peptide tachykinin NK3 receptor antagonist and it has a very high affinity for native guinea pig (pK(i) value 7.8) tachykinin NK(3...
Parathyroid hormone (1-34) (bovine)
Parathyroid hormone (1-34) (bovine) is a parathyroid hormone (PTH) receptor agonist. It increases calcium and inorganic phosphate levels in the serum of young r...
ML 349 is a lysophospholipase 2 inhibitor with IC50 value of 144 nM.
Bakuchiol is a phytoestrogen isolated from the seeds of Psoralea corylifolia L with an anti-tumor effects.
Isofagomine, an imino pyranose compound, has been found to be a glucosylceramidase stimulant and could exhibit activity in Gaucher's disease.
REP 3123 dihydrochloride
REP 3123 dihydrochloride is a selective inhibitor of methionyl-tRNA synthetase (MetRS) used as an antibiotic for the treatment of Clostridium difficile infectio...