PTAC oxalate - CAS 201939-40-4
Category: Inhibitor
Please be kindly noted products are not for therapeutic use. We do not sell to patients.
Molecular Formula:
C12H19N3S2.C2H2O4
Molecular Weight:
359.46
COA:
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Targets:
mAChR
Description:
PTAC oxalate is a muscarinic receptor ligand, which shows partial agonist activity at the M2 and M4 receptors, with minor antagonistic activity at m1, m3, m5 receptors (Ki values are 2.8, 0.2, 0.6, 0.2 and 0.8 nM respectively).
Purity:
≥98% by HPLC
Synonyms:
(1R,5R,6R)-6-[4-(Propylthio)-1,2,5-thiadiazol-3-yl]-1-azabicyclo[3.2.1]octane oxalate
Storage:
Store in a cool and dry place (or refer to the Certificate of Analysis).
MSDS:
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InChIKey:
LXXQOVMTAFXOKQ-IYPAPVHQSA-N
InChI:
InChI=1S/C12H19N3S2.C2H2O4/c1-2-6-16-12-11(13-17-14-12)10-8-15-5-3-4-9(10)7-15;3-1(4)2(5)6/h9-10H,2-8H2,1H3;(H,3,4)(H,5,6)/t9-,10-;/m0./s1
Canonical SMILES:
CCCSC1=NSN=C1C2CN3CCCC2C3.C(=O)(C(=O)O)O
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CAS 201939-40-4 PTAC oxalate

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