|Description||The deuterated labelled form of Ponatinib whichb is a novel, potent multi-target inhibitor of Abl, PDGFRα, VEGFR2, FGFR1 and Src with IC50 of 0.37 nM, 1.1 nM, 1.5 nM, 2.2 nM and 5.4 nM, respectively.|
|Related CAS||943319-70-8 (unlabelled)|
A labelled Naftifine, which is an allylamine antifungal drug for the topical treatment of tinea pedis, tinea cruris, and tinea corporis, probably involves selec...
Prothipendyl-D6-oxalate is a labelled salt of Prothipendyl. Prothipendyl is a weak dopamine receptor antagonist that is used to treat anxiety and agitation in p...
The deuterated labelled form ofPimozide (Orap) which is an antipsychotic drug of the diphenylbutylpiperidine class.
Ethacrynic acid-d5 is a deuterated ethacrynic acid used as an internal standard for GC- or LC-mass spectrometry.
A labelled Alosetrone. Alosetrone is a 5-HT3 antagonist indicated for diarrhea diarrhea caused by irritable bowel syndrome (IBS) in women.
2-Thiouracil-13C,15N2 is a labelled 2-Thiouracil. 2-Thiouracil is a thiolated uracil derivative that is a known antihyperthyroid agent.
An isotope labelled Sulfadiazine. Sulfadiazine is an antibiotic. It is commonly used to treat urinary tract infections and burns.
An isotope labelled Ethyl Maltol, which is an extract from medicinal plants such as P. Incarnata and can be used as an anticonvulsant, acting as a depressant, a...
An isotope labelled Stavudine. Stavudine is an antiretroviral medication used to prevent and treat HIV/AIDS.
An isotope labelled of Pentoxifylline. Pentoxifylline can be used for the treatment of muscle pain in people with peripheral artery disease.
Diazoxide-d3 is a labelled analogue of Diazoxide. Diazoxide is a potassium channel stimulator used as a vasodilator for acute hypertension.
Labelled Olmesartan, which is a specific angiotensin II type 1 (AT1) receptor antagonist with antihypertensive effect. hAT1 receptors: IC50 = 6.7 nM
Gepirone-d8 is a deuterated Gepirone. Gepirone is an antidepressant which is under development to treat depression and anxiety.
An isotope labelled Sulfasalazine. Sulfasalazine is a medication used to treat rheumatoid arthritis, ulcerative colitis, and Crohn's disease.
Labelled Oxaprozin, which is a inhibitor of both COX-1 and COX-2.
Lumefantrine D18 is the deuterium labeled Lumefantrine, which is an antimalarial drug.
Cycloguanil D6 is a deuterium labelled analogue of Cycloguanil. Cycloguanil is an inhibitor of dihydrofolate reductase and a metabolite of proguanil.
An isotope labelled of Sildenafil. Sildenafil can be usedto treat erectile dysfunction and pulmonary arterial hypertension.