|Description||The deuterated labelled form of Ponatinib whichb is a novel, potent multi-target inhibitor of Abl, PDGFRα, VEGFR2, FGFR1 and Src with IC50 of 0.37 nM, 1.1 nM, 1.5 nM, 2.2 nM and 5.4 nM, respectively.|
|Related CAS||943319-70-8 (unlabelled)|
An isotope labelled of Salicylic Acid. Salicylic Acid is an organic buliding block that can be used in organic synthesis.
Miglustat Hydrochloride-d9 is a labelled Miglustat Hydrochloride which is an inhibitor of a-glucosidase 1 as well as being an inhibitor of HIV cytopathicity.
A labelled Oxcarbazepine, which inhibits the binding of [3H]BTX to sodium channels with IC50 of 160 μM.
Sulfachloropyridazine-13C6 is an isotope labelled Sulfachloropyridazine, which is an antibiotic used for bacterial infections.
Griseofulvin-d3 is a labelled analogue of Griseofulvin. Griseofulvin is an antifungal drug used for the treatment of dermatophytoses and some other infections c...
Azelnidipine D7 is a labelled Azelnidipine. Azelnidipine is a calcium channel blocker with a hypotensive activity.
Ethopabate-D5 is a labelled Ethopabate, which is used as a coccidiostat in poultry.
The stable isotope labelled form of Haloperidol which could be an antipsychotic agent for blocking dopamine receptors.
Macitentan-d7 is a labelled Macitentan. Macitentan is an endothelin receptor antagonist (ERA) used for the treatment of pulmonary arterial hypertension (PAH).
One of the isotopic labelled form of Sunitinib, which is a receptor tyrosine kinases inhibitor.
An isotope labelled Sorafenib. Sorafenib is a small inhibitor of several tyrosine protein kinases, such as VEGFR, PDGFR and Raf family kinases, for the treatmen...
the labelled Lanthionine Ketimine-R-5-Ethyl Ester.
An isotope labelled of Cephalexin. Cephalexin is an antibiotic that can treat a number of bacterial infections.
An isotope labelled of Tiotropium bromide. Tiotropium bromide is an anticholinergic bronchodilator used in the management of chronic obstructive pulmonary disea...
Isotope labelled Eplerenone. Eplerenone is a potassium-sparing diuretic that selectively blocks aldosterone activation of the mineralcorticoid receptor, demonst...
A labelled Rilmenidine. Rilmenidine is a novel non-nucleoside reverse transcriptase inhibitor used as an anti-HIV agent. Rilpivirine seems to be well tolerated ...
Pirbuterol-D9 acetate is a labelled Pirbuterol acetate. Pirbuterol acetate is a short-acting β2 adrenoreceptor agonist.
Almotriptan-d6 Malate is a labelled Almotriptan. Almotriptan is a triptan medication used for the treatment of acute headaches including migraine headache.
Amitriptyline-d6 HCl is a labelled analogue of Amitriptyline. Amitriptyline is a psychotropic drug used for the treatment of major depression, anxiety and other...