PKR-IN-1 - CAS 1260075-17-9
Catalog number: B0084-463157
Category: Inhibitor
Please be kindly noted products are not for therapeutic use. We do not sell to patients.
Molecular Formula:
C24H26N4O3S
Molecular Weight:
450.55
COA:
Inquire
Targets:
Others
Description:
Activator of pyruvate kinase isoenzyme M2 (PKM2), an enzyme involved in glycolysis. Since all tumor cells exclusively express the embryonic M2 isoform of PK, it is hypothesized that PKM2 is a potential target for cancer therapy. Modulation of PKM2 might also be effective in the treatment of obesity, diabetes, autoimmune conditions, and antiproliferation-dependent diseases.
Ordering Information
Catalog Number Size Price Stock Quantity
B0084-463157 100 mg $599 In stock
Bulk Inquiry
Purity:
>98%
Synonyms:
PKR-IN-1
MSDS:
Inquire
InChIKey:
XAYGBKHKBBXDAK-UHFFFAOYSA-N
InChI:
InChI=1S/C24H26N4O3S/c29-24(28-15-13-27(14-16-28)17-18-6-7-18)20-8-10-21(11-9-20)26-32(30,31)22-5-1-3-19-4-2-12-25-23(19)22/h1-5,8-12,18,26H,6-7,13-17H2
Canonical SMILES:
C1CC1CN2CCN(CC2)C(=O)C3=CC=C(C=C3)NS(=O)(=O)C4=CC=CC5=C4N=CC=C5
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

Related Products


CAS 104206-65-7 Nitisinone

Nitisinone
(CAS: 104206-65-7)

Nitisinone(SC0735) is an inhibitor of the enzyme 4-hydroxyphenylpyruvate dioxygenase.

CAS 13422-55-4 Methylcobalamin

Methylcobalamin
(CAS: 13422-55-4)

Vitamin B12 (cobalamin) refers to a group of chemically-related cobalt containing molecules involved in cell processes such as DNA synthesis, fatty acid synthes...

CAS 1258275-73-8 TMPA

TMPA
(CAS: 1258275-73-8)

TMPA is an antagonist of nuclear receptor Nur77 (Kd = 1.45 ± 0.35 μM) and LKB1 interaction.

CAS 343306-71-8 Sugammadex

Sugammadex
(CAS: 343306-71-8)

Sugammadex, a modified γ-cyclodextrin, with a lipophilic core and a hydrophilic periphery, is an agent for reversal of neuromuscular blockade by the agent rocu...

CAS 34670-43-4 4-Azido-L-phenylalanine hydrochloride

4-Azido-L-phenylalanine hydrochloride
(CAS: 34670-43-4)

4-Azido-L-phenylalanine is an unnatural derivative of L-phenylalanine, a nonpolar, essential amino acid that naturally occurs in the human body and is also used...

CAS 107538-05-6 Dexmecamylamine

Dexmecamylamine
(CAS: 107538-05-6)

Dexmecamylamine is a nicotinic channel modulator with antidepressant activity. It demonstrated positive effects in a number of animal models of depression and a...

CAS 856676-23-8 Choline Fenofibrate

Choline Fenofibrate
(CAS: 856676-23-8)

Choline Fenofibrate is the choline salt of fenofibric acid under clinical development as a combination therapy with rosuvastatin for the management of dyslipide...

BMS-505130
(CAS: 468715-83-5)

BMS-505130 is a potent and selective serotonin transport inhibitor with K(i) of 0.18 nM.

Chemical Structure

CAS 1260075-17-9 PKR-IN-1

Quick Inquiry

Verification code

Featured Items