PHP 501 trifluoroacetate - CAS 1236105-75-1
Category: Inhibitor
Please be kindly noted products are not for therapeutic use. We do not sell to patients.
Molecular Formula:
C20H21N3O.CF3CO2H
Molecular Weight:
433.42
COA:
Inquire
Targets:
GABA Receptor
Description:
PHP 501 trifluoroacetate is potent GABAA antagonist (Ki = 0.0028 μM at rat GABAA receptors; IC50 = 0.024 μM at human α1β2γ2 GABAA-expressing tsA201 cells), without disrupting hGAT-1, hGAT-2, hGAT-3 or hBGT-1 GABA transporters.
Purity:
≥98% by HPLC
Synonyms:
PHP 501 trifluoroacetate; PHP501 trifluoroacetate; PHP-501 trifluoroacetate; 4-(5-[1,1'-Biphenyl]-3-yl-1-hydroxy-1H-pyrazol-4-yl)piperidine trifluoroacetate
Storage:
Store in a cool and dry place (or refer to the Certificate of Analysis).
MSDS:
Inquire
InChIKey:
SULXXKLCQRXMHP-UHFFFAOYSA-N
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

Related GABA Receptor Products


CAS 56776-32-0 Etifoxine Hydrochloride

Etifoxine Hydrochloride
(CAS: 56776-32-0)

Etifoxine Hydrochloride is Potentiator of GABAA receptor with anxiolytic and anticonvulsant activity.

CAS 951650-22-9 NS 11394

NS 11394
(CAS: 951650-22-9)

NS 11394 is a drug with selectivity for the α3 and α5 subtypes. It acts as a subtype-selective positive allosteric modulator at GABAA receptors. It is used as a...

CAS 138729-47-2 Eszopiclone

Eszopiclone
(CAS: 138729-47-2)

Eszopiclone is an active stereoisomer of zopiclone with hypnotic and sedative activity and without significant anxiolytic activity. Eszopiclone is a GABA A rece...

CAS 53552-05-9 (-)-Bicuculline methochloride

(-)-Bicuculline methochloride
(CAS: 53552-05-9)

(-)-Bicuculline methochloride is the methochloride salt of (+)-bicuculline, which is a potent antagonist of GABAA receptors.

CAS 21967-41-9 Baicalin

Baicalin
(CAS: 21967-41-9)

Baicalin is a flavone found in several species in the genus Scutellaria, including Scutellaria baicalensis and Scutellaria lateriflora. Baicalin is a positive a...

CAS 139667-74-6 CGP 52432

CGP 52432
(CAS: 139667-74-6)

CGP52432 is a potent and selective GABAB receptor antagonist with IC50 value of 85 nM.

CAS 152273-12-6 U-93631

U-93631
(CAS: 152273-12-6)

U 93631 is a ligand at the picrotoxin site of GABA(A) receptors, allosterically antagonizing GABA-induced Cl- currents. U-93631 causes rapid decay of gamma-amin...

CAS 96604-21-6 Ocinaplon

Ocinaplon
(CAS: 96604-21-6)

Ocinaplon is a GABAA receptor modulator and it can be used for the treatment of generalized anxiety disorder.

Chemical Structure

CAS 1236105-75-1 PHP 501 trifluoroacetate

Quick Inquiry

Verification code

Featured Items