Molecular Formula: | |
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Molecular Formula | C20H21N3O.CF3CO2H |
Molecular Weight: | |
Molecular Weight | 433.42 |
COA: | |
COA | Inquire |
Targets: | |
Targets | GABA Receptor |
Description: | |
Description | PHP 501 trifluoroacetate is potent GABAA antagonist (Ki = 0.0028 μM at rat GABAA receptors; IC50 = 0.024 μM at human α1β2γ2 GABAA-expressing tsA201 cells), without disrupting hGAT-1, hGAT-2, hGAT-3 or hBGT-1 GABA transporters. |
Purity: | |
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Purity | ≥98% by HPLC |
Synonyms: | |
Synonyms | PHP 501 trifluoroacetate; PHP501 trifluoroacetate; PHP-501 trifluoroacetate; 4-(5-[1,1'-Biphenyl]-3-yl-1-hydroxy-1H-pyrazol-4-yl)piperidine trifluoroacetate |
Storage: | |
Storage | Store in a cool and dry place (or refer to the Certificate of Analysis). |
MSDS: | |
MSDS | Inquire |
InChIKey: | |
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InChIKey | SULXXKLCQRXMHP-UHFFFAOYSA-N |
Chemical Structure