PHP 501 trifluoroacetate - CAS 1236105-75-1
Category: Inhibitor
Please be kindly noted products are not for therapeutic use. We do not sell to patients.
Molecular Formula:
C20H21N3O.CF3CO2H
Molecular Weight:
433.42
COA:
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Targets:
GABA Receptor
Description:
PHP 501 trifluoroacetate is potent GABAA antagonist (Ki = 0.0028 μM at rat GABAA receptors; IC50 = 0.024 μM at human α1β2γ2 GABAA-expressing tsA201 cells), without disrupting hGAT-1, hGAT-2, hGAT-3 or hBGT-1 GABA transporters.
Purity:
≥98% by HPLC
Synonyms:
PHP 501 trifluoroacetate; PHP501 trifluoroacetate; PHP-501 trifluoroacetate; 4-(5-[1,1'-Biphenyl]-3-yl-1-hydroxy-1H-pyrazol-4-yl)piperidine trifluoroacetate
Storage:
Store in a cool and dry place (or refer to the Certificate of Analysis).
MSDS:
Inquire
InChIKey:
SULXXKLCQRXMHP-UHFFFAOYSA-N
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CAS 1236105-75-1 PHP 501 trifluoroacetate

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