PHP 501 trifluoroacetate - CAS 1236105-75-1
Category: Inhibitor
Please be kindly noted products are not for therapeutic use. We do not sell to patients.
Molecular Formula:
C20H21N3O.CF3CO2H
Molecular Weight:
433.42
COA:
Inquire
Targets:
GABA Receptor
Description:
PHP 501 trifluoroacetate is potent GABAA antagonist (Ki = 0.0028 μM at rat GABAA receptors; IC50 = 0.024 μM at human α1β2γ2 GABAA-expressing tsA201 cells), without disrupting hGAT-1, hGAT-2, hGAT-3 or hBGT-1 GABA transporters.
Publication citing BOC Sciences Products
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4. Risk assessment of intake of pyrrolizidine alkaloids from herbal teas and medicines following realistic exposure scenarios
5. Machine learning models identify molecules active against the Ebola virus in vitro
6. Electrophotographic member, process cartridge and electrophotographic apparatus

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Purity:
≥98% by HPLC
Synonyms:
PHP 501 trifluoroacetate; PHP501 trifluoroacetate; PHP-501 trifluoroacetate; 4-(5-[1,1'-Biphenyl]-3-yl-1-hydroxy-1H-pyrazol-4-yl)piperidine trifluoroacetate
Storage:
Store in a cool and dry place (or refer to the Certificate of Analysis).
MSDS:
Inquire
InChIKey:
SULXXKLCQRXMHP-UHFFFAOYSA-N
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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Chemical Structure

CAS 1236105-75-1 PHP 501 trifluoroacetate

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