PF-4840154 - CAS 1332708-14-1
Catalog number: 1332708-14-1
Category: Inhibitor
Please be kindly noted products are not for therapeutic use. We do not sell to patients.
Molecular Formula:
C26H38N6O2
Molecular Weight:
466.62
COA:
Inquire
Targets:
TRP Channel
Description:
PF-4840154 has been foundd to be superior than Mustard Oil as a TrpA1 agonists. IC50: 97 nM and 23 nM (EC50) for hTrpA1 and rTrpA1 respectively.
Purity:
98%
Appearance:
Powder
Synonyms:
PF-4840154; PF 4840154; PF4840154. CHEMBL1818218; GTPL-6309; CS-5066; GTPL 6309; CS 5066; GTPL6309; CS5066; SCHEMBL17185544; BDBM50350947
Solubility:
10 mM in DMSO
Storage:
-20ºC Freeze
MSDS:
Inquire
Application:
PF-4840154 has been foundd to be superior than Mustard Oil as a TrpA1 agonists.
Shelf Life:
As supplied, 2 years from the QC date provided on the Certificate of Analysis, when stored properly
Quantity:
Milligrams-Grams
InChIKey:
PPANZCQXFYBGHN-UHFFFAOYSA-N
InChI:
InChI=1S/C26H38N6O2/c1-20(2)15-27-24-23(25(33)28-16-21-7-4-3-5-8-21)17-29-26(30-24)32-12-10-31(11-13-32)18-22-9-6-14-34-19-22/h3-5,7-8,17,20,22H,6,9-16,18-19H2,1-2H3,(H,28,33)(H,27,29,30)
Canonical SMILES:
CC(C)CNC1=NC(=NC=C1C(=O)NCC2=CC=CC=C2)N3CCN(CC3)CC4CCCOC4
Current Developer:
Pfizer
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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