PDK1 inhibitor 2610
Category: Inhibitor
Please be kindly noted products are not for therapeutic use. We do not sell to patients.
Molecular Formula:
C25H15N5.HCl
Molecular Weight:
421.88
COA:
Inquire
Targets:
PDK-1 | PI3K
Description:
PDK1 inhibitor 2610 is an ATP-competitive and selective dual PI3K and PDPK1 inhibitor (IC50 values 34 nM and 94 nM for PDK1 and p-T308-PKB, respectively).
Brife Description:
dual PI3K and PDPK1 inhibitor
Purity:
99%
MSDS:
Inquire
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

Related PDK-1 Products


LY-3023414
(CAS: 1386874-06-1)

LY3023414, a quinoline derivative, has been found to be a PI3Kα and mTOR inhibitor that could influence cell proliferation and cycle of tumor cells. It was just...

CAS 938444-93-0 D 106669

D 106669
(CAS: 938444-93-0)

D 106669 is a potent and selective PI3K inhibitor.

CAS 1180676-32-7 PS 48

PS 48
(CAS: 1180676-32-7)

PS 48 is an allosteric activator of phosphoinositide-dependent protein kinase 1 (PDPK1; PDK1) binding to the PIF-binding pocket of PDK1.

CAS 702674-56-4 BX912

BX912
(CAS: 702674-56-4)

BX-912 is a selective inhibitor of 3-Phosphoinositide-dependent Kinase-1 (PDK1) with IC50 of 12 nM; >10 fold selectivity over PKA, PKC, C-Kit, EGFR etc.

AM-8508
(CAS: 1338483-67-2)

AM-8508 is a selective Phosphatidylinositol-3-kinase delta (PI3Kδ) inhibitor. AM-8508 exhibits good cellular potency (in vitro pAKT IC50 = 4.6 nM ) and excellen...

CAS 702675-74-9 BX795

BX795
(CAS: 702675-74-9)

BX795 is a potent and selective inhibitor of PDK1, IKKε and TBK1, which regulates the production of Type 1 interferons during bacterial and viral infection. BX7...

CAS 1276110-06-5 HS-173

HS-173
(CAS: 1276110-06-5)

HS-173 is a potent and selective PI3Kα inhibitor displaying anticancer activity. HS-173 was shown to induce apoptosis via arresting the cell cycle at the G2/M p...

CAS 1032568-63-0 Copanlisib

Copanlisib
(CAS: 1032568-63-0)

Copanlisib is a phosphoinositide 3-kinase (PI3K) inhibitor with potential antineoplastic activity. BAY 80-6946 inhibits the activation of the PI3K signaling pat...

Quick Inquiry

Verification code

Featured Items