PDE1-IN-2 - CAS 1904611-63-7
Category: Inhibitor
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Molecular Formula:
C16H21BrN4O2
Molecular Weight:
381.27
COA:
Inquire
Targets:
Phosphodiesterase (PDE)
Description:
PDE1-IN-2 is an inhibitor of PDE1 that has IC50 values of 6, 140 and 164 nM for PDE1C, PDE1B and PDE1A, respectvely.
Brife Description:
An inhibitor of PDE1
Synonyms:
PDE1 IN 2; 6-bromo-7-(cyclopentylmethyl)-3-(oxan-4-yl)-[1,2,4]triazolo[4,3-a]pyrazin-8-one
Solubility:
DMSO: 10mM
Storage:
Store in a cool and dry place (or refer to the Certificate of Analysis).
MSDS:
Inquire
Boiling Point:
563.8±60.0 ℃ at 760 Torr
Density:
1.70±0.1 g/cm
InChIKey:
UDLAXUPVISWZSI-UHFFFAOYSA-N
InChI:
1S/C16H21BrN4O2/c17-13-10-21-14(12-5-7-23-8-6-12)18-19-15(21)16(22)20(13)9-11-3-1-2-4-11/h10-12H,1-9H2
Canonical SMILES:
C1CCC(C1)CN2C(=CN3C(=NN=C3C2=O)C4CCOCC4)Br
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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Chemical Structure

CAS 1904611-63-7 PDE1-IN-2

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