Palosuran - CAS 540769-28-6
Catalog number: B0084-182338
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C25H30N4O2
Molecular Weight:
418.54
COA:
Inquire
Targets:
Urotensin Receptor
Description:
Palosuran is a new Urotensin-II receptor antagonist (IC50=3.6±0.2 nM).
Ordering Information
Catalog Number Size Price Stock Quantity
B0084-182338 5 mg $179 In stock
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Publication citing BOC Sciences Products
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Purity:
≥95%
Appearance:
White to off-white Solid
Synonyms:
1-[2-(4-benzyl-4-hydroxypiperidin-1-yl)ethyl]-3-(2-methylquinolin-4-yl)urea; ACT-058362;
Solubility:
Soluble in DMSO
Storage:
Store at -20 °C
MSDS:
Inquire
Application:
Urotensin-II receptor antagonist
Quality Standard:
Enterprise Standard
Shelf Life:
As supplied, 2 years from the QC date provided on the Certificate of Analysis, when stored properly
Quantity:
Milligrams-Grams
InChIKey:
WYJCYXOCHXWTHG-UHFFFAOYSA-N
InChI:
1S/C25H30N4O2/c1-19-17-23(21-9-5-6-10-22(21)27-19)28-24(30)26-13-16-29-14-11-25(31,12-15-29)18-20-7-3-2-4-8-20/h2-10,17,31H,11-16,18H2,1H3,(H2,26,27,28,30)
Canonical SMILES:
CC1=NC2=CC=CC=C2C(=C1)NC(=O)NCCN3CCC(CC3)(CC4=CC=CC=C4)O
Current Developer:
Actelion Pharmaceuticals
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