Oxamflatin - CAS 151720-43-3
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C17H14N2O4S
Molecular Weight:
342.37
COA:
Inquire
Targets:
HDAC
Description:
Oxamflatin, also known as Metacept-3, an aromatic sulfonamide derivative, is a cell-permeable, potent HDAC inhibitor (IC50= 15.7 nM) with antitumor effect.
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Synonyms:
(E)-5-[3-(benzenesulfonamido)phenyl]-N-hydroxypent-2-en-4-ynamide; (2E)-5-(3-(phenylsulfonylamino)phenyl)pent-2-ene-4-ynohydroxamic acid; oxamflatin; Metacept-3
Solubility:
DMSO: ≥125 mg/mL
Storage:
Store in a cool and dry place (or refer to the Certificate of Analysis).
MSDS:
Inquire
Density:
1.44±0.1 g/cm3
InChIKey:
QRPSQQUYPMFERG-LFYBBSHMSA-N
InChI:
1S/C17H14N2O4S/c20-17(18-21)12-5-4-7-14-8-6-9-15(13-14)19-24(22,23)16-10-2-1-3-11-16/h1-3,5-6,8-13,19,21H,(H,18,20)/b12-5+
Canonical SMILES:
C1=CC=C(C=C1)S(=O)(=O)NC2=CC=CC(=C2)C#CC=CC(=O)NO
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CAS 151720-43-3 Oxamflatin

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