|Description||OTS-964, a thienoquinolin derivative, is a TOPK inhibitor and prabably be useful in studying anticancer agent as an analogue of OTS-514. It is still under preclinical trial. IC50: 28 nM.|
|Solubility||10 mM in DMSO|
|Application||OTS-964 is a TOPK inhibitor and prabably be useful in studying anticancer agent as an analogue of OTS-514.|
|Shelf Life||As supplied, 2 years from the QC date provided on the Certificate of Analysis, when stored properly|
|Current Developer||OncoTherapy Science; University of Chicago|
A synthetic analogue of α-melanocyte stimulating hormone (α-MSH)
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