|Targets||Neurokinin 1 Receptor|
|Description||Orvepitant is a potent and selective Neurokinin-1 (NK1) antagonist. It may be potential therapeutic for the treatment of patients with major depressive disorder (MDD), anxiety and insomnia. It was developed by GlaxoSmithKline and is in clinical phase 2 trials.|
|Solubility||Soluble in DMSO, not in water|
|Application||Orvepitant may be potential therapeutic for the treatment of patients with major depressive disorder (MDD), anxiety and insomnia.|
|Quality Standard||In-house standard|
|Boiling Point||627.5±55.0 °C | Condition: Press: 760 Torr|
|Density||1.37±0.1 g/cm3 | Condition: Temp: 20 °C Press: 760 Torr|
|Current Developer||Orvepitant was developed by GlaxoSmithKline and is in clinical phase 2 trials.|
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