ORM-15341 - CAS 1297537-33-7
Catalog number: 1297537-33-7
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C19H17ClN6O2
Molecular Weight:
396.83
COA:
Inquire
Targets:
Androgen Receptor
Description:
ORM-15341, an androgen receptor antagonist, could have potential effect against prostate cancer and commonly found as an active main metabolite of ODM-201. IC50: 38 nM.
Purity:
98%
Appearance:
Powder
Synonyms:
UNII-9EPS75QMTL; ORM-15341; 9EPS75QMTL; SCHEMBL1815556; GMBPVBVTPBWIKC-NSHDSACASA-N; CS-5191
Solubility:
DMSO: > 37 mg/mL
Storage:
-20ºC Freeze
MSDS:
Inquire
Application:
ORM-15341 is an androgen receptor antagonist that could have potential effect against prostate cancer and commonly found as an active main metabolite of ODM-201.
Shelf Life:
As supplied, 2 years from the QC date provided on the Certificate of Analysis, when stored properly
Quantity:
Milligrams-Grams
InChIKey:
GMBPVBVTPBWIKC-NSHDSACASA-N
InChI:
InChI=1S/C19H17ClN6O2/c1-11(22-19(28)18-8-17(12(2)27)23-24-18)10-26-6-5-16(25-26)13-3-4-14(9-21)15(20)7-13/h3-8,11H,10H2,1-2H3,(H,22,28)(H,23,24)/t11-/m0/s1
Canonical SMILES:
CC(CN1C=CC(=N1)C2=CC(=C(C=C2)C#N)Cl)NC(=O)C3=CC(=NN3)C(=O)C
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

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