|Targets||PDGFR | VEGFR|
|Description||TSU-68 (SU6668; Orantinib) is a novel multiple receptor tyrosine kinase inhibitor with IC50 of 2.1 μM, 8 nM and 1.2 μM for VEGF-R1, PDGF-Rβ and FGF-R1, respectively; has greatest potency against PDGFR autophosphorylation.|
|Synonyms||TSU-68; SU6668; NSC 702827.|
|Current Developer||Taiho Pharma Inc.|
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