Omaciclovir - CAS 124265-89-0
Catalog number:
124265-89-0
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C10H15N5O3
Molecular Weight:
253.26
COA:
Inquire
Targets:
DNA/RNA Synthesis
Description:
This active molecular is a DNA-directed DNA polymerase inhibitor potentially originated by Medivir AB. Omaciclovir can be selectively phosphorylated by viral thymidine kinase to its monophosphate form and it is further modified to a triphosphate, which is an inhibitor of VZV DNA polymerase. Preclinical trials for Herpes simplex virus infections, HIV infections and Varicella zoster virus infections were discontinued.
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Purity:
98%
Appearance:
Powder
Synonyms:
2-HMHBG; UNII-C9H909GLI3; Omaciclovir [USAN:INN]; C9H909GLI3; H 2G;2-amino-9-[(2R)-4-hydroxy-2-(hydroxymethyl)butyl]-3H-purin-6-one
Solubility:
Soluble in DMSO
Storage:
-20°C Freezer
MSDS:
Inquire
Application:
Herpes simplex virus infections, HIV infections and Varicella zoster virus infections
Quality Standard:
In-house standard
Shelf Life:
2 month in rt, long time
Quantity:
Milligrams-Grams
InChIKey:
SCBFBAWJWLXVHS-ZCFIWIBFSA-N
InChI:
InChI=1S/C10H15N5O3/c11-10-13-8-7(9(18)14-10)12-5-15(8)3-6(4-17)1-2-16/h5-6,16-17H,1-4H2,(H3,11,13,14,18)/t6-/m1/s1
Canonical SMILES:
C1=NC2=C(N1CC(CCO)CO)NC(=NC2=O)N
Current Developer:
Originator: Medivir AB
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