Olodaterol - CAS 868049-49-4
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C21H26N2O5
Molecular Weight:
386.44
COA:
Inquire
Targets:
Adrenergic Receptor
Description:
Olodaterol, also referred to BI1744, is a long acting β2-agonist (β2-ARs; EC50s = 97.7 and 2,725 nM for human β2- and β1-ARs, respectively) used as an inhalation for treating patients with chronic obstructive pulmonary disease (COPD), manufactured by Boehringer-Ingelheim.
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Brife Description:
A long acting beta-adrenoceptor agonist (EC50= 1.4±0.08 Nm)
Related CAS:
869477-96-3 (HCl)
Synonyms:
6-hydroxy-8-[(1R)-1-hydroxy-2-[[1-(4-methoxyphenyl)-2-methylpropan-2-yl]amino]ethyl]-4H-1,4-benzoxazin-3-one; 6-hydroxy-8-(1-hydroxy-2-((2-(4-methoxyphenyl)-1,1-dimethylethyl)amino)ethyl)-2H-1,4-benzoxazin-3(4H)-one; BI 1744 CL; BI-1744 CL; olodaterol; Striverdi; Respimat
Solubility:
H2O: 6.2 mg/mL
Storage:
Store in a cool and dry place (or refer to the Certificate of Analysis).
MSDS:
Inquire
Boiling Point:
649.0±55.0 ℃ at 760 Torr
Density:
1.250±0.06 g/cm3
InChIKey:
COUYJEVMBVSIHV-SFHVURJKSA-N
InChI:
1S/C21H26N2O5/c1-21(2,10-13-4-6-15(27-3)7-5-13)22-11-18(25)16-8-14(24)9-17-20(16)28-12-19(26)23-17/h4-9,18,22,24-25H,10-12H2,1-3H3,(H,23,26)/t18-/m0/s1
Canonical SMILES:
CC(C)(CC1=CC=C(C=C1)OC)NCC(C2=CC(=CC3=C2OCC(=O)N3)O)O
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CAS 868049-49-4 Olodaterol

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