Odelepran - CAS 676501-25-0
Catalog number: 676501-25-0
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C20H24FN3O3
Molecular Weight:
373.43
COA:
Inquire
Targets:
Opioid Receptor
Description:
Odelepran is a opioid receptor antagonist. It is used for the treatment of alcohol dependence. It was developed by Lilly and was in clinical phase 2 trial, but now it is terminated.
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Purity:
98%
Appearance:
Solid powder
Synonyms:
Ondelopran;6-[2-Fluoro-4-[[2-(oxan-4-yl)ethylamino]methyl]phenoxy]pyridine-3-carboxamide;LY2196044;LY-2196044
Solubility:
Soluble in DMSO, not in water
Storage:
-20°C Freezer
MSDS:
Inquire
Application:
Odelepran is used for the treatment of alcohol dependence.
Quality Standard:
In-house standard
Quantity:
Milligrams-Grams
Boiling Point:
525.2±50.0 °C | Condition: Press: 760 Torr
Density:
1.213±0.06 g/cm3 | Condition: Temp: 20 °C Press: 760 Torr
InChIKey:
QWNDOCKIKKQJNN-UHFFFAOYSA-N
InChI:
InChI=1S/C20H24FN3O3/c21-17-11-15(12-23-8-5-14-6-9-26-10-7-14)1-3-18(17)27-19-4-2-16(13-24-19)20(22)25/h1-4,11,13-14,23H,5-10,12H2,(H2,22,25)
Canonical SMILES:
C1COCCC1CCNCC2=CC(=C(C=C2)OC3=NC=C(C=C3)C(=O)N)F
Current Developer:
Odelepran was developed by Lilly and was in clinical phase 2 trial, but now it is terminated.
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