Odelepran - CAS 676501-25-0
Catalog number: 676501-25-0
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
Molecular Weight:
Opioid Receptor
Odelepran is a opioid receptor antagonist. It is used for the treatment of alcohol dependence. It was developed by Lilly and was in clinical phase 2 trial, but now it is terminated.
Publictions citing BOC Sciences Products
  • >> More
Solid powder
Soluble in DMSO, not in water
-20°C Freezer
Odelepran is used for the treatment of alcohol dependence.
Quality Standard:
In-house standard
Boiling Point:
525.2±50.0 °C | Condition: Press: 760 Torr
1.213±0.06 g/cm3 | Condition: Temp: 20 °C Press: 760 Torr
Canonical SMILES:
Current Developer:
Odelepran was developed by Lilly and was in clinical phase 2 trial, but now it is terminated.
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

Related Opioid Receptor Products

(CAS: 854601-70-0)

Naloxegol is a CYP3A4 enzyme inhibitor. It is also a peripherally-selective opioid antagonist. It is used as the treatment of opioid-induced constipation. lt is...

CAS 156727-74-1 SNC 80

SNC 80
(CAS: 156727-74-1)

SNC 80 is a potent and non-peptide δ-opioid agonist, displaying 2000-fold selectivity over μ-opioid receptors. SNC 80 exhibits antinociceptive as well as pro-co...

CAS 67197-96-0 (±)-U-50488 hydrochloride

(±)-U-50488 hydrochloride
(CAS: 67197-96-0)

(±)-U-50488 hydrochloride is a selective κ-opioid agonist with no μ-opioid antagonist effects. (±)-U-50488 hydrochloride blocks Na+ channels at high concentrati...

CAS 1216621-00-9 Trap 101

Trap 101
(CAS: 1216621-00-9)

Trap 101 is a potent and selective nociceptin/orphanin FQ (NOP) receptor antagonist (pA2 = 7.75) with selectivity for NOP receptors over classical opioid recept...

CAS 115199-84-3 ICI 199,441 hydrochloride

ICI 199,441 hydrochloride
(CAS: 115199-84-3)

ICI 199,441 hydrochloride is the hydrochloride salt of ICI 199,441, which is a selective and highly potent κ agonist. It is 146-fold more active than U-50488 in...

(CAS: 1401028-24-7)

TRV130 is an oxaspiro compound that has been found to be a μ-opioid receptor G protein ligand and could be used in pain therapy. IC50: 8.1 (pEC50. G protein ass...

CAS 213130-17-7 [Phe1Ψ(CH2-NH)Gly2]Nociceptin(1-13)NH2

(CAS: 213130-17-7)

[Phe1Ψ(CH2-NH)Gly2]Nociceptin(1-13)NH2 is the first selective antagonist to prevent the binding of the endogenous ligand orphanin FQ​/Nociceptin (OFQ​/N) at the...

CAS 152657-84-6 Nalfurafine

(CAS: 152657-84-6)

Nalfurafine is a selective and centrally-penetrant κ-opioid receptor (KOR) agonist without significant activity on μ- and δ-opioid receptors. With antipruritic ...

(CAS: 1346133-08-1)

LY2795050, a κ-opioid Receptor antagonist, has been found to be effective in imaging KOR behaving as a PET tracer. IC50: 0.72 nM and 25.8 nM for κ-opioid Recept...

CAS 189388-22-5 Endomorphin 1

Endomorphin 1
(CAS: 189388-22-5)

Endomorphin 1 is a high affinity (Ki = 360 pM) and highly selective agonist of theμ-opioid receptor with 4000- and 15000-fold preference over δ and κ respective...

(CAS: 519052-02-9)

CP866087 is a selective mu-opioid receptor antagonist.

CAS 133267-27-3 Fedotozine tartrate

Fedotozine tartrate
(CAS: 133267-27-3)

Fedotozine tartrate is a kappa(1a) opioid receptor agonist.

CAS 178803-51-5 SNC 162

SNC 162
(CAS: 178803-51-5)

SNC 162 is a potent and selective non-peptide δ-opioid receptor agonist (Ki = 0.63 nM), displaying > 8000-fold selectivity over μ-opioid receptors. SNC 162 is c...

6'-GNTI dihydrochloride

6'-GNTI dihydrochloride is a potent and selective κ/δ-opioid heterodimer receptor agonist (EC50 = 39.8, 112.5 and > 1000 nM for κ/δ, κ/μ and δ/μ, respectively) ...

(CAS: 475150-69-7)

BAN ORL 24, a spiro-isobenzofuran compound, has been found to be a NOP receptor antagonist and could be used to restrain the reduction of locomotor motions with...

CAS 34552-83-5 Loperamide HCl

Loperamide HCl
(CAS: 34552-83-5)

Loperamide HCl is an opioid-receptor agonist with an ED50 of 0.15 mg/kg.

CAS 83335-41-5 Dynorphin B

Dynorphin B
(CAS: 83335-41-5)

Dynorphin B is a 13-residue opioid peptide, which is derived from the cleavage of prodynorphin and found widely distributed in the central nervous system. It ac...

CAS 684238-37-7 BMS 986187

BMS 986187
(CAS: 684238-37-7)

BMS 986187 is a potent and selective δ-opioid receptor positive allosteric modulator (EC50 = 30 nM) exhibiting 100-fold selectivity for δ over μ-opioid receptor...

CAS 357-08-4 Naloxone hydrochloride

Naloxone hydrochloride
(CAS: 357-08-4)

Naloxone HCl is an opioid inverse agonist drug used to counter the effects of opiate overdose.

CAS 152685-85-3 Hemorphin-7

(CAS: 152685-85-3)

Hemorphin-7, a hemorphin peptide with antinociceptive and antihypertensive effects, is an endogenous opioid peptide derived from the β-chain of hemoglobin. Hemo...

Quick Inquiry

Verification code

Featured Items