NVP-BGJ398 phosphate - CAS 1310746-10-1
Catalog number: 1310746-10-1
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C26H34Cl2N7O7P
Molecular Weight:
658.47
COA:
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Targets:
FGFR
Description:
Potent and selective inhibitor of fibroblast growth factor receptor (FGFR) tyrosine kinases 1, 2, 3 and 4 (with IC50 values of 0.9, 1.4, 1.0 and 60 nM for FGFR1, FGFR2, FGFR3, and FGFR4 respectively); it showed siginificant antitumor activity in RT112 bladder cancer xenografts models overexpressing wild-type FGFR3.
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Purity:
>98%
Synonyms:
Infigratinib phosphate; BGJ-398 phosphate
MSDS:
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CAS 1310746-10-1 NVP-BGJ398 phosphate

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