NVP-BAG956 - CAS 853910-02-8
Catalog number:
853910-02-8
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C28H21N5
Molecular Weight:
427.5
COA:
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Targets:
PDK-1
Description:
NVP-BAG956 is a potent, ATP-competitive and selective dual PI3K and PDK1 inhibitor in vitro and in vivo. It inhibits cellular AKT phosphorylation at Thr308 and blocks cell proliferation, causing arrest in G1 phase of the cell cycle. It slows tumor progression in mouse xenograft models.
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Purity:
>98%
Synonyms:
BAG 956
MSDS:
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Chemical Structure

CAS 853910-02-8 NVP-BAG956

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