Nuvenzepine - CAS 96487-37-5
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C19H20N4O2
Molecular Weight:
336.39
COA:
Inquire
Targets:
mAChR
Description:
Nuvenzepine, a new pirenzepine-analog, is an mAChR antagonist, administered intraduodenally, displayed a long-lasting and dose-dependent inhibition of neostigmine-induced intestinal motility in anaesthetized cats.
Publictions citing BOC Sciences Products
  • >> More
Synonyms:
11-(1-methylpiperidine-4-carbonyl)-6H-pyrido[3,2-c][1,5]benzodiazepin-5-one; 11-(N-methylisonipecotyl)-6,11-dihydro-5H-pyrido(2,3-b)(1,5)benzodiazepin-5-one; DF 545; DF-545; nuvenzepine
Storage:
Store in a cool and dry place (or refer to the Certificate of Analysis).
MSDS:
Inquire
Boiling Point:
522.3±50.0 ℃ at 760 Torr
Density:
1.267±0.06 g/cm3
InChIKey:
HPKYRXAEGNUARA-UHFFFAOYSA-N
InChI:
1S/C19H20N4O2/c1-22-11-8-13(9-12-22)19(25)23-16-7-3-2-6-15(16)21-18(24)14-5-4-10-20-17(14)23/h2-7,10,13H,8-9,11-12H2,1H3,(H,21,24)
Canonical SMILES:
CN1CCC(CC1)C(=O)N2C3=CC=CC=C3NC(=O)C4=C2N=CC=C4
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

Related mAChR Products


CAS 62-97-5 Diphemanil Methylsulfate

Diphemanil Methylsulfate
(CAS: 62-97-5)

Diphemanil Methylsulfate is a quaternary ammonium anticholinergic.It binds muscarinic acetycholine receptors (mAchR).

CAS 3254-89-5 Diphenidol hydrochloride

Diphenidol hydrochloride
(CAS: 3254-89-5)

Diphenidol HCl is a potent antagonist of muscarinic M2 and M3 receptor with pKb of 6.72 and 7.02, respectively, used in the treatment of vomiting and vertigo.

CAS 1159101-48-0 Tarafenacin D-tartrate

Tarafenacin D-tartrate
(CAS: 1159101-48-0)

Tarafenacin is a highly selective M3 muscarinic receptor antagonist (Ki=0.19 nM), ~200 fold selectivity over M2 receptor.

CAS 125-53-1 oxyphencyclimine

oxyphencyclimine
(CAS: 125-53-1)

Oxyphencyclimine is a muscarinic cholinergic receptor antagonist and trade name is called as Daricon. Now it is applicated for the treatment of peptic ulcers an...

CAS 634616-95-8 TBPB

TBPB
(CAS: 634616-95-8)

TBPB is an allosteric M1 mAChR agonist that regulates amyloid processing and produces antipsychotic-like activity in rats.

CAS 96487-37-5 Nuvenzepine

Nuvenzepine
(CAS: 96487-37-5)

Nuvenzepine, a new pirenzepine-analog, is an mAChR antagonist, administered intraduodenally, displayed a long-lasting and dose-dependent inhibition of neostigmi...

CAS 131986-45-3 Xanomeline

Xanomeline
(CAS: 131986-45-3)

Xanomeline is a Muscarinic M1 and M4 receptor agonist under the development of Eli Lilly, though it is also known to act as a M5 receptor antagonist. Xanomeline...

CAS 54-71-7 Pilocarpine Hydrochloride

Pilocarpine Hydrochloride
(CAS: 54-71-7)

Pilocarpine HCl is a nonselective muscarinic acetylcholine receptor agonist used to produce an experimental model of epilepsy.

CAS 60-31-1 Acetylcholine Chloride

Acetylcholine Chloride
(CAS: 60-31-1)

Acetylcholine is an organic molecule that acts as a neurotransmitter in many organisms, including humans.

CAS 148-72-1 pilocarpine nitrate

pilocarpine nitrate
(CAS: 148-72-1)

pilocarpine nitrate is a non-selective muscarinic receptor agonist that can be used to treat glaucoma.

CAS 180468-39-7 Solifenacin hydrochloride

Solifenacin hydrochloride
(CAS: 180468-39-7)

Muscarinic M3 receptor antagoinst. Used in treatment of urinary incontinence.

CAS 1135242-13-5 VU 0357017 hydrochloride

VU 0357017 hydrochloride
(CAS: 1135242-13-5)

The hydrochloride salt form of VU0357017 which is a selective M1 agonists and has been found to be probably effective in the treatment of hippocampal-dependent ...

CAS 146422-58-4 CDD0102

CDD0102
(CAS: 146422-58-4)

CDD0102 is a selective M1 agonist which stimulated the secretion of APP from CHO-K1 cells expressing M1 receptors and penetrated into the brain following i.p. a...

CI 969
(CAS: 113590-49-1)

This active molecular is a muscarinic agonist agent.

CAS 385367-47-5 Tarafenacin

Tarafenacin
(CAS: 385367-47-5)

Tarafenacin is a highly selective M3 muscarinic receptor antagonist. It was the most potent in inhibiting carbachol-induced bladder contractions of the anti-ch...

CAS 84504-69-8 Irsogladine maleate

Irsogladine maleate
(CAS: 84504-69-8)

Irsogladine is a PDE4 inhibitor and muscarinic acetylcholine receptor binder. It inhibits bFGF-induced angiogenesis in wild-type, tPA-knockout, and uPA-knockout...

PQCA
(CAS: 1144504-35-7)

This active molecular is a muscarinic M1 receptor positive allosteric modulator which is able to improve cognitive measures in rat and rhesus monkeys. PQCA is v...

CAS 55-48-1 Atropine sulfate

Atropine sulfate
(CAS: 55-48-1)

Atropine is is a naturally occurring tropane alkaloid extracted from deadly nightshade acts as a competitive muscarinic acetylcholine receptor antagonist.

CAS 68252-19-7 Pirmenol

Pirmenol
(CAS: 68252-19-7)

Pirmenol, also known as CI-845, a new antiarrhythmic drug, inhibits muscarinic acetylcholine receptor-operated K+ current in the guinea pig heart. However, pirm...

CAS 155-41-9 Methscopolamine

Methscopolamine
(CAS: 155-41-9)

Methscopolamine is a muscarinic acetylcholine receptor blocker.

Chemical Structure

CAS 96487-37-5 Nuvenzepine

Quick Inquiry

Verification code

Featured Items