Nuvenzepine - CAS 96487-37-5
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C19H20N4O2
Molecular Weight:
336.39
COA:
Inquire
Targets:
mAChR
Description:
Nuvenzepine, a new pirenzepine-analog, is an mAChR antagonist, administered intraduodenally, displayed a long-lasting and dose-dependent inhibition of neostigmine-induced intestinal motility in anaesthetized cats.
Publictions citing BOC Sciences Products
  • >> More
Synonyms:
11-(1-methylpiperidine-4-carbonyl)-6H-pyrido[3,2-c][1,5]benzodiazepin-5-one; 11-(N-methylisonipecotyl)-6,11-dihydro-5H-pyrido(2,3-b)(1,5)benzodiazepin-5-one; DF 545; DF-545; nuvenzepine
Storage:
Store in a cool and dry place (or refer to the Certificate of Analysis).
MSDS:
Inquire
Boiling Point:
522.3±50.0 ℃ at 760 Torr
Density:
1.267±0.06 g/cm3
InChIKey:
HPKYRXAEGNUARA-UHFFFAOYSA-N
InChI:
1S/C19H20N4O2/c1-22-11-8-13(9-12-22)19(25)23-16-7-3-2-6-15(16)21-18(24)14-5-4-10-20-17(14)23/h2-7,10,13H,8-9,11-12H2,1H3,(H,21,24)
Canonical SMILES:
CN1CCC(CC1)C(=O)N2C3=CC=CC=C3NC(=O)C4=C2N=CC=C4
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

Related mAChR Products


CAS 96487-37-5 Nuvenzepine

Nuvenzepine
(CAS: 96487-37-5)

Nuvenzepine, a new pirenzepine-analog, is an mAChR antagonist, administered intraduodenally, displayed a long-lasting and dose-dependent inhibition of neostigmi...

PQCA
(CAS: 1144504-35-7)

This active molecular is a muscarinic M1 receptor positive allosteric modulator which is able to improve cognitive measures in rat and rhesus monkeys. PQCA is v...

CAS 124937-52-6 Tolterodine tartrate

Tolterodine tartrate
(CAS: 124937-52-6)

Tolterodine has a high affinity and specificity for muscarinic receptors in vitro and it exhibits selectivity for the urinary bladder over salivary glands in vi...

CAS 320345-99-1 Aclidinium Bromide

Aclidinium Bromide
(CAS: 320345-99-1)

Aclidinium Bromide(LAS 34273; LAS-W 330) is a long-acting, inhaled muscarinic antagonist as a maintenance treatment for chronic obstructive pulmonary disease (C...

CAS 6989-98-6 Tubocurarine hydrochloride pentahydrate

Tubocurarine hydrochloride pentahydrate
(CAS: 6989-98-6)

Tubocurarine is a toxic alkaloid. It is an acetylcholine receptor (AChR)-blocking agent. Tubocurarine is now rarely used as an adjunct for clinical anesthesia b...

CAS 55-48-1 Atropine sulfate

Atropine sulfate
(CAS: 55-48-1)

Atropine is is a naturally occurring tropane alkaloid extracted from deadly nightshade acts as a competitive muscarinic acetylcholine receptor antagonist.

CAS 10405-02-4 Trospium chloride

Trospium chloride
(CAS: 10405-02-4)

Trospium chloride is a competitive muscarinic cholinergic receptor antagonist.

CAS 514-65-8 Biperiden

Biperiden
(CAS: 514-65-8)

Biperiden is an antiparkinsonian agent, which is the selective central M1 cholinoreceptors blocker. It is used for the adjunctive treatment of all forms of Park...

CAS 286930-03-8 Fesoterodine Fumarate

Fesoterodine Fumarate
(CAS: 286930-03-8)

Fesoterodine Fumarate is an antimuscarinic agent and is rapidly de-esterified to its active metabolite 5-hydroxymethyl tolterodine that is a muscarinic receptor...

CAS 54-71-7 Pilocarpine Hydrochloride

Pilocarpine Hydrochloride
(CAS: 54-71-7)

Pilocarpine HCl is a nonselective muscarinic acetylcholine receptor agonist used to produce an experimental model of epilepsy.

CAS 129-77-1 Piperidolate hydrochloride

Piperidolate hydrochloride
(CAS: 129-77-1)

The hydrochloride salt form of Piperidolate which is an antimuscarinic and could restrain the abnormal activity caused by acetylcholine.

CAS 60-31-1 Acetylcholine Chloride

Acetylcholine Chloride
(CAS: 60-31-1)

Acetylcholine is an organic molecule that acts as a neurotransmitter in many organisms, including humans.

CAS 62-97-5 Diphemanil Methylsulfate

Diphemanil Methylsulfate
(CAS: 62-97-5)

Diphemanil Methylsulfate is a quaternary ammonium anticholinergic.It binds muscarinic acetycholine receptors (mAchR).

CAS 5908-99-6 Atropine sulfate salt monohydrate

Atropine sulfate salt monohydrate
(CAS: 5908-99-6)

Atropine is a competitive muscarinic acetylcholine receptor antagonist with an IC50 of 2.5 nM.

CAS 84504-69-8 Irsogladine maleate

Irsogladine maleate
(CAS: 84504-69-8)

Irsogladine is a PDE4 inhibitor and muscarinic acetylcholine receptor binder. It inhibits bFGF-induced angiogenesis in wild-type, tPA-knockout, and uPA-knockout...

CAS 107233-08-9 Cevimeline

Cevimeline
(CAS: 107233-08-9)

Cevimeline is a selective M1 receptor agonist.

CAS 1227923-29-6 MK-7622

MK-7622
(CAS: 1227923-29-6)

MK-7622 is a cholinesterase inhibitor under evaluation for the treatment of Alzheimer's disease. No studies have been published on this compound in the peer-rev...

CAS 146422-58-4 CDD0102

CDD0102
(CAS: 146422-58-4)

CDD0102 is a selective M1 agonist which stimulated the secretion of APP from CHO-K1 cells expressing M1 receptors and penetrated into the brain following i.p. a...

CAS 141064-23-5 Xanomeline oxalate

Xanomeline oxalate
(CAS: 141064-23-5)

Muscarinic receptors are G protein-coupled acetylcholine receptors that play diverse roles. Xanomeline oxalate is a potent agonist of muscarinic acetylcholine r...

CAS 1098-97-1 Pyrithioxin

Pyrithioxin
(CAS: 1098-97-1)

Pyrithioxin, a pyridine thiol derivatives, could be used in the treatment of traumatic brain injury sequelae and some sorts of cerebral infarct patients with He...

Chemical Structure

CAS 96487-37-5 Nuvenzepine

Quick Inquiry

Verification code

Featured Items