|Description||Nuvenzepine, a new pirenzepine-analog, is an mAChR antagonist, administered intraduodenally, displayed a long-lasting and dose-dependent inhibition of neostigmine-induced intestinal motility in anaesthetized cats.|
|Synonyms||11-(1-methylpiperidine-4-carbonyl)-6H-pyrido[3,2-c][1,5]benzodiazepin-5-one; 11-(N-methylisonipecotyl)-6,11-dihydro-5H-pyrido(2,3-b)(1,5)benzodiazepin-5-one; DF 545; DF-545; nuvenzepine|
|Storage||Store in a cool and dry place (or refer to the Certificate of Analysis).|
|Boiling Point||522.3±50.0 ℃ at 760 Torr|
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Diphenidol HCl is a potent antagonist of muscarinic M2 and M3 receptor with pKb of 6.72 and 7.02, respectively, used in the treatment of vomiting and vertigo.
Tarafenacin is a highly selective M3 muscarinic receptor antagonist (Ki=0.19 nM), ~200 fold selectivity over M2 receptor.
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Acetylcholine is an organic molecule that acts as a neurotransmitter in many organisms, including humans.
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Muscarinic M3 receptor antagoinst. Used in treatment of urinary incontinence.
VU 0357017 hydrochloride
The hydrochloride salt form of VU0357017 which is a selective M1 agonists and has been found to be probably effective in the treatment of hippocampal-dependent ...
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This active molecular is a muscarinic agonist agent.
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