NSC 663284 - CAS 383907-43-5
Category:
Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C15H16ClN3O3
Molecular Weight:
321.76
COA:
Inquire
Targets:
Others
Description:
NSC 663284 is a potent, irreversible, cell permeable and mixed competitive Cdc25 dual specificity phosphatases inhibitor (IC50= 0.21 μM), and poorly inhibits other phosphatases, including Vaccinia virus VH1-related (IC50 = 4.0 μM), PTP1B (no inhibition), and the mitogen-activated protein kinase phosphatases (MKP) MKP-1 or -3 (no inhibition).
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Synonyms:
6-chloro-7-(2-morpholin-4-ylethylamino)quinoline-5,8-dione; NSC 663284; NSC-663284; NSC663284
Solubility:
DMSO: ≥150 mg/mL
Storage:
Store in a cool and dry place (or refer to the Certificate of Analysis).
MSDS:
Inquire
Boiling Point:
478.8±45.0 ℃ at 760 Torr
Density:
1.41±0.1 g/cm3
InChIKey:
BMKPVDQDJQWBPD-UHFFFAOYSA-N
InChI:
1S/C15H16ClN3O3/c16-11-13(18-4-5-19-6-8-22-9-7-19)15(21)12-10(14(11)20)2-1-3-17-12/h1-3,18H,4-9H2
Canonical SMILES:
C1COCCN1CCNC2=C(C(=O)C3=C(C2=O)N=CC=C3)Cl
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CAS 383907-43-5 NSC 663284

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