|Description||Neostigmine is a parasympathomimetic compound, which acts as a reversible acetylcholinesterase inhibitor. It is used in the treatment of myasthenia gravis, ogilvie syndrome and urinary retention without the presence of a blockage. It is also used to reverse the effects of muscle relaxants such as gallamine and tubocurarine. It is in the cholinergic family of medications and works by blocking the action of acetylcholinesterase and therefore increases the levels of acetylcholine. It does not cross the blood-brain barrier.|
|Synonyms||CCRIS 3079; CCRIS3079; CCRIS-3079; 3-[[(Dimethylamino)carbonyl]oxy]-N,N,N-trimethylbenzenaminium;Eustigmin;Eustigmine;Vagostigmine;Prostigmin;Polstigmine|
|Solubility||Soluble in DMSO, not in water|
|Application||Neostigmine is used in the treatment of myasthenia gravis, ogilvie syndrome and urinary retention without the presence of a blockage. It is also used to reverse the effects of muscle relaxants such as gallamine and tubocurarine.|
|Quality Standard||In-house standard|
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