Nelotanserin - CAS 839713-36-9
Catalog number: 839713-36-9
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C18H15BrF2N4O2
Molecular Weight:
437.24
COA:
Inquire
Targets:
5-HT Receptor
Description:
Nelotanser is Serotonin 2A receptor inverse agonist. In Aug 2016, Axovant Sciences initiated a phase-II clinical trial in Lewy body disease in USA.
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Purity:
98%
Appearance:
Powder
Synonyms:
1-[3-(4-bromo-2-methylpyrazol-3-yl)-4-methoxyphenyl]-3-(2,4-difluorophenyl)urea;APD 125
Solubility:
DMSO: ≥ 32 mg/mL
Storage:
-20℃ Freezer
MSDS:
Inquire
Application:
Lewy body disease
Quality Standard:
In-house standard
Shelf Life:
2 month in rt, long time
Quantity:
Milligrams-Grams
InChIKey:
COSPVUFTLGQDQL-UHFFFAOYSA-N
InChI:
InChI=1S/C18H15BrF2N4O2/c1-25-17(13(19)9-22-25)12-8-11(4-6-16(12)27-2)23-18(26)24-15-5-3-10(20)7-14(15)21/h3-9H,1-2H3,(H2,23,24,26)
Canonical SMILES:
CN1C(=C(C=N1)Br)C2=C(C=CC(=C2)NC(=O)NC3=C(C=C(C=C3)F)F)OC
Current Developer:
Arena Pharmaceuticals; Axovant Sciences
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CAS 839713-36-9 Nelotanserin

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