Nelotanserin - CAS 839713-36-9
Catalog number: 839713-36-9
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
Molecular Weight:
5-HT Receptor
Nelotanser is Serotonin 2A receptor inverse agonist. In Aug 2016, Axovant Sciences initiated a phase-II clinical trial in Lewy body disease in USA.
Publictions citing BOC Sciences Products
  • >> More
1-[3-(4-bromo-2-methylpyrazol-3-yl)-4-methoxyphenyl]-3-(2,4-difluorophenyl)urea;APD 125
DMSO: ≥ 32 mg/mL
-20℃ Freezer
Lewy body disease
Quality Standard:
In-house standard
Shelf Life:
2 month in rt, long time
Canonical SMILES:
Current Developer:
Arena Pharmaceuticals; Axovant Sciences
Molecular Weight Calculator Molarity Calculator Solution Dilution Calculator

Related 5-HT Receptor Products

CAS 97469-12-0 α-Methyl-5-hydroxytryptamine maleate

α-Methyl-5-hydroxytryptamine maleate
(CAS: 97469-12-0)

α-Methyl-5-hydroxytryptamine maleate, a salt of α-Methylserotonin maleate, is a 5-HT2B receptor selective agonist with pKi values of 8.4, 6.1 and 7.3 at 5-HT2B,...

CAS 137403-12-4 L-694,247

(CAS: 137403-12-4)

L-694,247 is a highly selective and extremely potent 5-HT1D receptor agonist.

CAS 213007-95-5 Org 37684

Org 37684
(CAS: 213007-95-5)

Org 37684 is a 5-HT2C receptor agonist.

CAS 66611-27-6 RU 24969 hemisuccinate

RU 24969 hemisuccinate
(CAS: 66611-27-6)

RU 24969 hemisuccinate is a potent and selective agonist at the 5-HT1A and 5-HT1B receptors. It is centrally active following systemic administration.

Lasmiditan hydrochloride
(CAS: 613677-28-4)

Lasmiditan hydrochloride is a potent and selective 5-HT1F receptor agonist that can be used for the treatment of acute migraine.

CAS 190508-50-0 AT 1015

AT 1015
(CAS: 190508-50-0)

AT 1015 has been found to be a 5-HT2A receptor antagonist and exhibit antithrombotic activities.

CAS 148672-15-5 GMC 2-29

GMC 2-29
(CAS: 148672-15-5)

GMC 2-29 is a potent and selective 5-HT1B/1D antagonist.

CAS 179756-85-5 Eptapirone

(CAS: 179756-85-5)

Eptapirone, a triazine derivative, has been found to be a 5-HT1A receptor agonist and was once studied as an antidepressant agent. pKi: 8.33.

CAS 64887-14-5 Urapidil HCl

Urapidil HCl
(CAS: 64887-14-5)

Urapidil HCl is a hydrochloride salt form of urapidil which is α1-adrenoceptor antagonist and 5-HT1A receptor agonist with pIC50 of 6.13 and 6.4 respectively.

CAS 210821-63-9 Org 12962 hydrochloride

Org 12962 hydrochloride
(CAS: 210821-63-9)

Org 12962 hydrochloride is a 5-HT2C receptor agonist with pEC50 value of 7.01. It shows antiaversive effects in the anxiety models in rats.

CAS 13523-86-9 Pindolol

(CAS: 13523-86-9)

Pindolol, an Indole derivative, could be used in the treatment of hypertension and arrhythmia for acting as a 5-HT1A/1B receptor antagonist. IC50: 33nM(Ki).

CAS 17375-63-2 BGC 20-761

BGC 20-761
(CAS: 17375-63-2)

BGC 20-761 is a selective, high affinity 5-HT6 antagonist (Ki = 20 nM). BGC 20-761 was shown to reverse the amnesic effects of scopolamine and enhance memory co...

CAS 58-39-9 Perphenazine

(CAS: 58-39-9)

Perphenazine is a typical antipsychotic. a piperazinyl phenothiazine, used to treat psychosis

CAS 101303-98-4 Zacopride hydrochloride

Zacopride hydrochloride
(CAS: 101303-98-4)

Zacopride hydrochloride is a highly potent 5-HT3 receptor antagonist (Ki = 0.38 nM) and 5-HT4 receptor agonist (Ki = 373 nM). Zacopride hydrochloride acts as an...

BMS 181101
(CAS: 146479-45-0)

BMS 181101, an indole derivative, has been found to be a 5-HT receptor agonist that could be probably effective against depression and also restrain serotonin r...

CAS 63687-94-5 GMC 1-116

GMC 1-116
(CAS: 63687-94-5)

GMC 1-116 is a metabolite of clozapine with weak 5-HT2 affinity and high M1 affinity (IC50 = 27 nM).

CAS 186826-17-5 ML 10302 hydrochloride

ML 10302 hydrochloride
(CAS: 186826-17-5)

ML 10302 hydrochloride is a 5-HT4 agonist with EC50 value of 4 nM. It can increase sAPPα levels in the cortex in an animal model of Alzheimer's disease and exhi...

CAS 145202-66-0 Rizatriptan Benzoate

Rizatriptan Benzoate
(CAS: 145202-66-0)

Rizatriptan Benzoate is a 5-HT1 agonist triptan drug for the treatment of migraine headaches.

CAS 5189-11-7 Pizotifen Malate

Pizotifen Malate
(CAS: 5189-11-7)

Pizotifen Malate is a benzocycloheptane based agent used for recurrent migraine headaches.

CAS 160521-72-2 BW 723C86 hydrochloride

BW 723C86 hydrochloride
(CAS: 160521-72-2)

BW 723C86 hydrochloride is a selective 5-HT2B receptor agonist used for the treatment of certain CNS disorders, such as epilepsy, migraine and feeding disorders...

Chemical Structure

CAS 839713-36-9 Nelotanserin

Quick Inquiry

Verification code

Featured Items