|Description||Nelotanser is Serotonin 2A receptor inverse agonist. In Aug 2016, Axovant Sciences initiated a phase-II clinical trial in Lewy body disease in USA.|
|Solubility||DMSO: ≥ 32 mg/mL|
|Application||Lewy body disease|
|Quality Standard||In-house standard|
|Shelf Life||2 month in rt, long time|
|Current Developer||Arena Pharmaceuticals; Axovant Sciences|
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Rupatadine inhibits both platelet-activating factor (PAF) and histamine (H1) effects through its interaction with specific receptors.
desmethyl-WAY 100635 trihydrochloride
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Way 100135 is a selective 5-HT1A receptor antagonist originated by Wyeth with IC50 value of 15 nM. IC 50 values for 5-HT1B, 1C, 2,α1, α2 and D2 receptors are ov...
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Lu AE58054 HCl salt
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LY 334370 hydrochloride
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CP 809101 hydrochloride
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NPEC-caged serotonin is a caged version of serotonin.
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LY 344864 racemate
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