|Description||Nedaplatin is a derivative of cisplatin and DNA damage agent for tumor colony forming units with IC50 of 94 μM.|
GRGDSPK, a linear integrin binding peptide, is an inhibitory peptide for RGD-mediated adhesion between integrin and extracellular matrix molecules.
CI 600 is a bio-active chemical, but no detailed information has been published yet.
Iopamidol is a nonionic, low-osmolar iodinated contrast agent, developed by Bracco.
Rafigrelide is a platelet aggregation inhibitor, which plays a central role in atherothrombotic events. It could prolonge clot formation time and reduce clot st...
Lificiguat, also known as YC-1, is a inhibitor of Hypoxia-inducible factor-1alpha (HIF-1alpha). YC-1 is widely used as a potent inhibitor of HIF-1alpha both in ...
Triacetin, an non-ionic surfactant, could be widely used because of its characteristics like dispersion, emulsification and solubilization capacity. The FEMA nu...
The D-Tartrate salt form of Isofagomine, an imino pyranose compound, has been found to be a glucosylceramidase stimulant and could exhibit activity in Gaucher's...
kb-NB77-78 is an analog of CID797718, which is a by-product of the synthesis of the parental compound, CID755673(PKD1 inhibitor).
Denatonium benzoate is a stimulant of the bitter taste receptors used as aversive agents (bitterants) to prevent inappropriate ingestion.
OTS-964, a thienoquinolin derivative, is a TOPK inhibitor and prabably be useful in studying anticancer agent as an analogue of OTS-514. It is still under precl...
CB-839 an is orally bioavailable inhibitor of glutaminase, with potential antineoplastic activity. Upon oral administration, CB-839 selectively and irreversibly...
AX-024 hydrochloride is an inhibitor of T cell receptor (TCR) that selectively inhibits the TCR-Nck interaction. By modulating TCR signaling, AX-024 prevents th...
LB-100 is a water solubleprotein phosphatase 2A (PP2A)inhibitor(IC50= 0.85 μM and 3.87 μM in BxPc-3 and Panc-1 cells) and enhanced the effects of sorafenib in H...
Botanical Source from Bufo bufo gargarizans and Bufo formosus, used for microbial transformation.
GSK-1268992 is one of a metabolite of Pazopanib which is a selective multi-targeted receptor tyrosine kinase inhibitor that blocks tumour growth and inhibits an...
MI-538, a 4-methylpyrazole compound, is a double substituted analogue with methylpyrazole at R1 and hydroxyl at R4. MI-538, a potent and selective MLL (Mixed Li...
(+)-Cloprostenol isopropyl ester
(+)-Cloprostenol isopropyl ester is a derivative of cloprostenol which has been found to be a FP receptor agonist as well as a luteolytic agent and could be use...
BMS-505130 is a potent and selective serotonin transport inhibitor with K(i) of 0.18 nM.
CS-M1996 is a 4′-Azidocytidine analogue. It can inhibit Hepatitis C virus replication.
PFK15 is a potent and selective 6-phosphofructo-2-kinase (PFKFB3) with IC50 of 207 nM.