|Description||Nebivolol selectively inhibits β1-adrenoceptor with IC50 of 0.8 nM.|
Prazosin HCl, a quinazoline derivative, is the first of a new chemical class of antihypertensives.
Isoetarine is a selective adrenergic beta-2 agonist. It is used as fast acting bronchodilator for emphysema, bronchitis and asthma. It has been listed.
Vilanterol, also known as GW-642444, is a long-acting beta-2 agonist drug, which in May 2013 was approved in combination with fluticasone furoate for sale as Br...
Fiduxosin hydrochloride is an alpha(1)-adrenoceptor antagonist used for the treatment of benign prostatic hyperplasia.
Phenylephrine HCl is a selective α1-adrenergic receptor agonist of the phenethylamine class used primarily as a decongestant, as an agent to dilate the pupil, a...
Salbutamol Sulfate is a Non-selective 2-adrenergic receptor agonist (IC50=8.93 µM)
Terazosin, works by blocking the action of adrenaline on smooth muscle of the bladder and the blood vessel walls, is a selective alpha1-antagonist used for trea...
Xylometazoline is an α-adrenoceptor agonist commonly used as nasal decongestant, exhibits highest potency at α2B-adrenoceptor subtype with EC50 of 99 μM.
Phentolamine Mesylate is a nonselective alpha-adrenergic antagonist with IC50 of 0.1 μM.
Mirabegron (formerly YM-178, trade name Myrbetriq) is a drug for the treatment of overactive bladder. It was developed by Astellas Pharma and was approved in th...
Terbutaline Sulfate is a selective β2-adrenergic receptor agonist with IC50 of 53 nM, used as a "reliever" inhaler in the management of asthma symptoms and as a...
Octopamine hydrochloride is an α-adrenoceptor agonist.
Hoku 81 is a bronchodilator, and one of the metabolites of tulobuterol.
Esmolol is a cardioselective beta1 receptor blocker with rapid onset, a very short duration of action, and no significant intrinsic sympathomimetic or membrane ...
The hydrochloride of Nifenalol. Nifenalol is a beta-adrenoceptor antagonist used for the treatment of cardiovascular and cerebrovascular diseases such as hypert...
Labetalol HCl is a dual antagonist for both selective alpha1-adrenergic and nonselective beta-adrenergic receptors, used in the treatment of high blood pressure...
Metoprolol succinate is a selective β-adrenoceptor antagonist. It is used in treatment of several diseases of the cardiovascular system. It is a drug used in th...
Bopindolol Malonate is a potent, non-selective, long-acting beta adrenoceptor antagonist. It demonstrates inhibition of H2O2-induced lipid peroxdiation. It is a...
Bometolol is a beta-adrenergic blocking drug.
Levosalbutamol tartrate, the R-enantiomer of salbutamol, is a short-acting β2 adrenergic receptor agonist used in the treatment of asthma and chronic obstructiv...