Nav1.7-IN-2 - CAS 1332295-35-8
Catalog number: 1332295-35-8
Category: Inhibitor
Not Intended for Therapeutic Use. For research use only.
Molecular Formula:
C22H22FN5O2
Molecular Weight:
407.44
COA:
Inquire
Targets:
Sodium Channel
Description:
Nav1.7-IN-2, a voltage-gated sodium channels, could be probably effective in chronic pain therapy. IC50: 80 nM.
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Purity:
98%
Appearance:
Powder
Synonyms:
Benzamide, 3-[[4-[3-(4-fluoro-2-methylphenoxy)-1-azetidinyl]-2-pyrimidinyl]amino]-N-methyl-
Solubility:
10 mM in DMSO
Storage:
-20ºC Freeze
MSDS:
Inquire
Application:
Nav1.7-IN-2 is a voltage-gated sodium channels and could be probably effective in chronic pain therapy.
Shelf Life:
As supplied, 2 years from the QC date provided on the Certificate of Analysis, when stored properly
Quantity:
Milligrams-Grams
InChIKey:
MFAKJGXMORSMIX-UHFFFAOYSA-N
InChI:
InChI=1S/C22H22FN5O2/c1-14-10-16(23)6-7-19(14)30-18-12-28(13-18)20-8-9-25-22(27-20)26-17-5-3-4-15(11-17)21(29)24-2/h3-11,18H,12-13H2,1-2H3,(H,24,29)(H,25,26,27)
Canonical SMILES:
CC1=C(C=CC(=C1)F)OC2CN(C2)C3=NC(=NC=C3)NC4=CC=CC(=C4)C(=O)NC
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